SCHEMBL24713404

SCHEMBL24713404

CN(C)/C=N/Sc1cc(NC(=O)OC(C)(C)C)cc2cnc(Cl)cc12

nearest known ligand 0.35

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MAPKAPK2 P49137 7/20 0.35
ALDH1A1 P00352 1/20 0.34
DGAT1 O75907 1/20 0.33
MAP4K4 O95819 1/20 0.33
ATR Q13535 1/20 0.32
TOP2A P11388 1/20 0.32
TOP2B Q02880 1/20 0.32
SYK P43405 1/20 0.32
GSK3B P49841 1/20 0.32
DYRK1A Q13627 1/20 0.32
CA12 O43570 1/20 0.31
CA1 P00915 1/20 0.31
CA9 Q16790 1/20 0.31
NAMPT P43490 1/20 0.31
AAK1 Q2M2I8 1/20 0.31
SREBF2 Q12772 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23619996 0.81 MAPKAPK2 (0.35) MAPKAPK2ALDH1A1DGAT1MAP4K4ATR
SCHEMBL24714003 0.81 ATR (0.42) MAPKAPK2ALDH1A1MAP4K4ATRTOP2A
SCHEMBL23619769 0.79 KCNJ5 (0.41) ALDH1A1
SCHEMBL23619944 0.75
SCHEMBL23620175 0.75
SCHEMBL23619734 0.67 NAMPT (0.39) ALDH1A1DGAT1TOP2ATOP2BSYK
SCHEMBL1368674 0.67 S1PR2 (0.58) MAPKAPK2MAP4K4ATRTOP2ATOP2B
SCHEMBL17336621 0.66 TRPV1 (0.46) MAPKAPK2ALDH1A1ATRSYKGSK3B
SCHEMBL10288086 0.66 GSK3B (0.54) MAPKAPK2MAP4K4ATRSYKGSK3B
SCHEMBL20525207 0.64 MAPKAPK2 (0.40) MAPKAPK2DGAT1MAP4K4ATRTOP2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4079724-A1 FUSED RING COMPOUND AND APPLICATION THEREOF Wuhan LL Science and Technology Development Co., Ltd. (CN) 2022-10-26 EP disclosed