SCHEMBL24722778

SCHEMBL24722778

CCOC(=O)c1cc(C(F)(F)F)c2c(n1)CN(C(=O)OC(C)(C)C)CC2

nearest known ligand 0.48

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 2/20 0.48
PARP1 P09874 1/20 0.42
TNKS2 Q9H2K2 1/20 0.42
PARP2 Q9UGN5 1/20 0.42
MTOR P42345 2/20 0.40
RAF1 P04049 1/20 0.39
BRAF P15056 1/20 0.39
ESR2 Q92731 1/20 0.39
NR1H2 P55055 1/20 0.38
F12 P00748 1/20 0.38
MAPT P10636 2/20 0.37
P2RX7 Q99572 2/20 0.37
GPR119 Q8TDV5 4/20 0.36
MEN1 O00255 1/20 0.36
ALDH1A1 P00352 1/20 0.36
HPGD P15428 1/20 0.36
KMT2A Q03164 1/20 0.36
TP53 P04637 1/20 0.35
POLB P06746 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23198443 0.88 ADORA1 (0.52) ADORA1PARP1TNKS2PARP2MTOR
SCHEMBL23199090 0.87 ADORA1 (0.51) ADORA1PARP1TNKS2PARP2MTOR
SCHEMBL23200226 0.86 ADORA1 (0.53) ADORA1PARP1TNKS2PARP2MTOR
SCHEMBL17551377 0.86 ADORA1 (0.50) ADORA1PARP1TNKS2PARP2MTOR
SCHEMBL24758537 0.86 ADORA1 (0.50) ADORA1PARP1TNKS2PARP2MTOR
SCHEMBL24759062 0.84 ADORA1 (0.48) ADORA1PARP1TNKS2PARP2MTOR
SCHEMBL23198536 0.81 ADORA1 (0.49) ADORA1PARP1TNKS2PARP2MTOR
SCHEMBL23199070 0.81 ADORA1 (0.46) ADORA1PARP1TNKS2PARP2MTOR
SCHEMBL17541080 0.81 GRM2 (0.50) ADORA1PARP1TNKS2PARP2
SCHEMBL19932597 0.81 ADORA1 (0.44) ADORA1PARP1TNKS2PARP2MTOR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20220402917-A1 COMPOUND AS SMALL MOLECULE INHIBITOR PD-1/PD-L1 AND APPLICATION THEREOF MEDSHINE DISCOVERY INC. (CN) 2022-12-22 US disclosed
EP-4043461-A1 COMPOUND AS SMALL MOLECULE INHIBITOR PD-1/PD-L1 AND APPLICATION THEREOF Medshine Discovery Inc. (CN) 2022-08-17 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20220402917-A1 COMPOUND AS SMALL MOLECULE INHIBITOR PD-1/PD-L1 AND APPLICATION THEREOF CD274, PDCD1, PDCD1LG2 ADORA1 2762/4885PARP1 342/4885TNKS2 1486/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.