SCHEMBL24729370

SCHEMBL24729370

O=C(O)c1ccc2sc(NC(=O)c3cc(F)c(F)c(F)c3)nc2c1

nearest known ligand 0.56

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.53
RAB9A P51151 3/20 0.53
KDM4E B2RXH2 1/20 0.53
NFKB1 P19838 1/20 0.53
HTT P42858 1/20 0.53
NFKB2 Q00653 1/20 0.53
RELA Q04206 1/20 0.53
TOP1 P11387 2/20 0.52
HSD17B10 Q99714 2/20 0.52
SMN1; SMN2 Q16637 2/20 0.51
MEN1 O00255 1/20 0.51
KMT2A Q03164 1/20 0.51
LRRK2 Q5S007 2/20 0.51
SCD O00767 2/20 0.50
HSD17B1 P14061 1/20 0.50
HSD17B2 P37059 1/20 0.50
DYRK1A Q13627 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29947576 1.00 NPC1 (0.53) NPC1RAB9AKDM4ENFKB1HTT
SCHEMBL24729347 0.90 HSD17B10 (0.64) NPC1RAB9AKDM4ENFKB1HTT
SCHEMBL29947591 0.90 HSD17B10 (0.64) NPC1RAB9AKDM4ENFKB1HTT
SCHEMBL24729516 0.87 NPC1 (0.54) NPC1RAB9AKDM4ENFKB1HTT
SCHEMBL29947476 0.85 HSD17B10 (0.50) NPC1RAB9AKDM4ENFKB1HTT
SCHEMBL24729247 0.85 HSD17B10 (0.50) NPC1RAB9AKDM4ENFKB1HTT
SCHEMBL29947662 0.84 HTT (0.61) NPC1RAB9AKDM4EHTTHSD17B10
SCHEMBL24729368 0.84 HTT (0.61) NPC1RAB9AKDM4EHTTHSD17B10
SCHEMBL24729361 0.82 NPC1 (0.61) NPC1RAB9AKDM4ENFKB1HTT
SCHEMBL24730598 0.82 NPC1 (0.53) NPC1RAB9AKDM4ENFKB1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022240213-A1 NOVEL BENZOTHIAZOLE DERIVATIVE, PREPARATION METHOD THEREFOR, AND USE THEREOF FOR PREVENTION OR TREATMENT OF LIVER DISEASE 에이치케이이노엔 주식회사 2022-11-17 WO disclosed