SCHEMBL24769192

SCHEMBL24769192

CCOc1cnc(Cl)cc1-c1cc(C)ncc1C(=O)OC

nearest known ligand 0.64

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
POLQ O75417 19/20 0.64
TDP1 Q9NUW8 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24500339 0.89 POLQ (0.61) POLQ
SCHEMBL30640125 0.89 POLQ (0.61) POLQ
SCHEMBL24769580 0.88 POLQ (0.60) POLQ
SCHEMBL24770165 0.85 POLQ (0.53) POLQ
SCHEMBL30017601 0.84 POLQ (0.64) POLQTDP1
SCHEMBL24770230 0.84 POLQ (0.64) POLQTDP1
SCHEMBL30858982 0.84 POLQ (0.54) POLQ
SCHEMBL30640105 0.83 POLQ (0.48) POLQ
SCHEMBL24769264 0.83 POLQ (0.48) POLQ
SCHEMBL24770191 0.83 POLQ (0.50) POLQ

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4352055-A1 O-LINKED THIADIAZOLYL COMPOUNDS AS DNA POLYMERASE THETA INHIBITORS Ideaya Biosciences, Inc. (US) 2024-04-17 EP disclosed
WO-2022259204-A1 O-LINKED THIADIAZOLYL COMPOUNDS AS DNA POLYMERASE THETA INHIBITORS IDEAYA BIOSCIENCES, INC. (US) 2022-12-15 WO disclosed
WO-2022259204-A1 O-LINKED THIADIAZOLYL COMPOUNDS AS DNA POLYMERASE THETA INHIBITORS IDEAYA BIOSCIENCES, INC. (US) 2022-12-15 WO disclosed