SCHEMBL24786151

SCHEMBL24786151

Cc1c(-n2cnc(C(=O)Cl)c2)ccc(Cl)c1F

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 2/20 0.41
KDM4E B2RXH2 1/20 0.35
LRRK2 Q5S007 1/20 0.33
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
NPC1 O15118 2/20 0.32
RAB9A P51151 2/20 0.32
SMN1; SMN2 Q16637 2/20 0.32
MAPT P10636 1/20 0.32
HPGD P15428 1/20 0.32
KCNH2 Q12809 3/20 0.31
SLC6A9 P48067 2/20 0.31
MAPK7 Q13164 1/20 0.31
GPR142 Q7Z601 1/20 0.31
PSEN1 P49768 1/20 0.30
PSEN2 P49810 1/20 0.30
APH1B Q8WW43 1/20 0.30
NCSTN Q92542 1/20 0.30
APH1A Q96BI3 1/20 0.30
PSENEN Q9NZ42 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18330395 0.89 KDM4E (0.46) NOTUMKDM4E
SCHEMBL18330398 0.80 PSEN1 (0.33) NOTUMPSEN1PSEN2APH1BNCSTN
SCHEMBL24786148 0.75 NOTUM (0.40) NOTUMKDM4EMEN1KMT2ASMN1; SMN2
SCHEMBL20176167 0.73 KDM4E (0.40) NOTUMKDM4E
SCHEMBL21004930 0.73 NOTUM (0.41) NOTUMKDM4E
SCHEMBL15933311 0.71 NOTUM (0.42) NOTUMKDM4E
SCHEMBL21901788 0.70 LRRK2 (0.37) KDM4ELRRK2NPC1RAB9ASMN1; SMN2
SCHEMBL14692532 0.69 KDM4E (0.48) NOTUMKDM4E
SCHEMBL15933233 0.69 NOTUM (0.39) NOTUMKDM4EMEN1KMT2ANPC1
SCHEMBL14692396 0.69 NOTUM (0.59) NOTUMMEN1KMT2ANPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3868753-B1 FACTOR XIA MACROCYCLIC INHIBITORS BEARING A NON-AROMATIC P2' GROUP BRISTOL MYERS SQUIBB CO (US) 2022-12-21 EP disclosed