Novobiocin

Novobiocin

SCHEMBL24805

CO[C@@H]1[C@@H](OC(N)=O)[C@@H](O)[C@H](Oc2ccc3c(O)c(NC(=O)c4ccc(O)c(CC=C(C)C)c4)c(=O)oc3c2C)OC1(C)C

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

gyrAgyrB

The experimentally established mechanism targets of Novobiocin. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 5/20 1.00
HSP90AB1 P08238 5/20 1.00
MAP1LC3B Q9GZQ8 2/20 1.00
MAP1LC3A Q9H492 2/20 1.00
POLQ O75417 1/20 1.00
ALB P02768 1/20 1.00
KDR P35968 1/20 1.00
ABCG2 Q9UNQ0 1/20 1.00
LMNA P02545 1/20 0.87
KDM4E B2RXH2 1/20 0.87
POLB P06746 1/20 0.73
MAPT P10636 1/20 0.73
RECQL P46063 1/20 0.73
NPSR1 Q6W5P4 1/20 0.73
ELAVL1 Q15717 1/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Novobiocin SCHEMBL14418054 1.00 HSP90AA1 (1.00) HSP90AA1HSP90AB1MAP1LC3BMAP1LC3APOLQ
Novobiocin SCHEMBL12077083 1.00 HSP90AA1 (1.00) HSP90AA1HSP90AB1MAP1LC3BMAP1LC3APOLQ
Novobiocin SCHEMBL16801983 1.00 HSP90AA1 (1.00) HSP90AA1HSP90AB1MAP1LC3BMAP1LC3APOLQ
Novobiocin SCHEMBL12967913 1.00 HSP90AA1 (1.00) HSP90AA1HSP90AB1MAP1LC3BMAP1LC3APOLQ
Novobiocin SCHEMBL24229298 1.00 HSP90AA1 (1.00) HSP90AA1HSP90AB1MAP1LC3BMAP1LC3APOLQ
Novobiocin SCHEMBL15314954 1.00 HSP90AA1 (1.00) HSP90AA1HSP90AB1MAP1LC3BMAP1LC3APOLQ
Novobiocin SCHEMBL24589148 1.00 HSP90AA1 (1.00) HSP90AA1HSP90AB1MAP1LC3BMAP1LC3APOLQ
Novobiocin SCHEMBL24336906 1.00 HSP90AA1 (1.00) HSP90AA1HSP90AB1MAP1LC3BMAP1LC3APOLQ
Novobiocin SCHEMBL23416512 1.00 HSP90AA1 (1.00) HSP90AA1HSP90AB1MAP1LC3BMAP1LC3APOLQ
Novobiocin SCHEMBL22023678 1.00 HSP90AA1 (1.00) HSP90AA1HSP90AB1MAP1LC3BMAP1LC3APOLQ

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 12539 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12622975-B2 Peptide-conjugated prodrugs BRANDEIS UNIVERSITY (US) 2026-05-12 US claimed
US-12624127-B2 Chitosan derivatives as antimicrobials and synergistic combinations thereof NANYANG TECHNOLOGICAL UNIVERSITY (SG) 2026-05-12 US claimed
EP-3790536-B1 NANOCONTAINERS FOR TRANSPORTING NONPOLAR, LIPOPHILIC SUBSTANCES SUCH AS ANTIBIOTICS KARLSRUHER INST TECHNOLOGIE (DE) 2026-04-22 EP claimed
US-20260091127-A1 JANUS PARTICLE-EMBEDDED MATERIALS FOR ANTIMICROBIAL APPLICATIONS UNIV INDIANA TRUSTEES (US) 2026-04-02 US claimed
EP-4683630-A1 VPS4B INHIBITOR FOR USE IN METHODS FOR THE TREATMENT OF HRD CANCER Institut Curie (FR) 2026-01-28 EP claimed
EP-4646432-A1 ANTI-IL-18BP ANTIBODIES Lassen Therapeutics, Inc. (US) 2025-11-12 EP claimed
EP-4646433-A1 ANTI-IL-18BP ANTIBODIES Lassen Therapeutics, Inc. (US) 2025-11-12 EP claimed
WO-2025224715-A1 METHODS FOR IMPROVING PRECISE GENOME MODIFICATION AND REDUCING UNWANTED MUTATIONS BY CRISPR-CAS EDITING KING ABDULLAH UNIVERISTY OF SCIENCE AND TECHNOLOGY (SA) 2025-10-30 WO claimed
US-20250263799-A1 METHODS OF TREATING CANCER USING REPLICATION STRESS MODULATORS THE INSTITUTE OF CANCER RES ROYAL CANCER HOSPITAL (GB) 2025-08-21 US claimed
US-12377052-B2 Dual-responsive nanoparticles for enhanced antibacterial efficacy WISCONSIN ALUMNI RESEARCH FOUNDATION (US) 2025-08-05 US claimed
EP-0025698-B1 CONTROLLED RELEASE FORMULATIONS ELI LILLY AND COMPANY (US) 1984-06-13 EP claimed
EP-0058867-A1 Method of producing a tricalcium phosphate bone ceramic for application as a bone implant, especially to fill cavities or for setting bone fractures in place after fracture, and tricalcium phosphate ceramic shaped articles produced according to this method mundipharma GmbH (DE) 1982-09-01 EP claimed
EP-0046270-A1 Novel derivatives of bio-affecting phenolic compounds and pharmaceutical composition containing them INTERx RESEARCH CORPORATION (US) 1982-02-24 EP claimed
US-4304855-A Allylic methyl-hydroxylated novobiocins THE UPJOHN COMPANY (US) 1981-12-08 US claimed
US-4293539-A Controlled release formulations and method of treatment ELI LILLY AND COMPANY (US) 1981-10-06 US claimed
US-4289757-A TOPICAL APPLICATION OF ANTIBIOTICS THE UPJOHN COMPANY (US) 1981-09-15 US claimed
US-4288543-A SAMPLING IN LIQUID PHASE WITH ANTIGROWTH AGENTS-BIOLOGICAL PFIZER INC. (US) 1981-09-08 US claimed
EP-0025698-A2 Controlled release formulations ELI LILLY AND COMPANY (US) 1981-03-25 EP claimed
US-4191740-A Synthetic resin-base, antibiotic compositions containing amino acids MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1980-03-04 US claimed
US-3932615-A Process for the preparation of granules MEIJI SEIKA CO., LTD. (JA) 1976-01-13 US claimed