SCHEMBL24812401

SCHEMBL24812401

C[C@@H]1COCCN1c1nc(-c2cccc3[nH]ccc23)nc2cc(C3CCCN3)[nH]c12

nearest known ligand 0.60

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ATR Q13535 15/20 0.60
BRAF P15056 1/20 0.58
PIK3CA P42336 4/20 0.55
MTOR P42345 4/20 0.55
PIK3CD O00329 1/20 0.55
CYP2D6 P10635 1/20 0.55
CYP2C9 P11712 1/20 0.55
PIK3CG P48736 1/20 0.55
ATRIP Q8WXE1 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24812407 0.89 ATR (0.65) ATRBRAFPIK3CAMTORPIK3CD
SCHEMBL24811616 0.81 ATR (0.71) ATRBRAFPIK3CAMTORPIK3CD
SCHEMBL24811195 0.81 ATR (0.57) ATRBRAFATRIP
SCHEMBL24810115 0.80 ATR (0.58) ATRBRAFPIK3CAMTORPIK3CD
SCHEMBL24812436 0.79 ATR (0.56) ATRBRAFATRIP
SCHEMBL24811608 0.78 ATR (0.67) ATRBRAFPIK3CAMTORPIK3CD
SCHEMBL24811617 0.78 ATR (0.80) ATRBRAFATRIP
SCHEMBL24811614 0.77 ATR (0.73) ATRBRAFMTORATRIP
SCHEMBL29805950 0.77 ATR (0.73) ATRBRAFMTORATRIP
SCHEMBL24811619 0.76 ATR (0.70) ATRBRAFATRIP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022268025-A1 ATR INHIBITOR AND USE THEREOF 成都苑东生物制药股份有限公司 2022-12-29 WO disclosed