SCHEMBL24823940

SCHEMBL24823940

CSn1ccc2cncnc21

nearest known ligand 0.42

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MKNK2 Q9HBH9 8/20 0.42
MKNK1 Q9BUB5 2/20 0.38
EGFR P00533 9/20 0.34
CYP1A2 P05177 2/20 0.32
CYP3A4 P08684 2/20 0.32
TSHR P16473 1/20 0.32
CLK4 Q9HAZ1 1/20 0.32
ALDH1A1 P00352 1/20 0.32
CYP2C9 P11712 1/20 0.32
HSD17B10 Q99714 1/20 0.32
PRMT5 O14744 1/20 0.31
WDR77 Q9BQA1 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30694603 0.75 MKNK2 (0.45) MKNK2MKNK1EGFRCYP1A2CYP3A4
SCHEMBL30564558 0.71 NOTUM (0.43) MKNK2MKNK1CYP1A2CYP3A4TSHR
SCHEMBL22622580 0.71 MKNK2 (0.45) MKNK2MKNK1EGFRCYP1A2CYP3A4
SCHEMBL13616341 0.71 MKNK2 (0.45) MKNK2MKNK1EGFRCYP1A2CYP3A4
SCHEMBL27821267 0.71 MKNK2 (0.45) MKNK2MKNK1EGFRCYP1A2CYP3A4
SCHEMBL6364432 0.70 MKNK2 (0.42) MKNK2MKNK1EGFR
SCHEMBL5068124 0.70 MKNK2 (0.42) MKNK2MKNK1EGFRCYP1A2CYP3A4
SCHEMBL5021603 0.70 MKNK2 (0.42) MKNK2MKNK1EGFRCYP1A2CYP3A4
SCHEMBL4417290 0.69 MKNK2 (0.41) MKNK2MKNK1EGFRCYP1A2CYP3A4
SCHEMBL29665757 0.69 MKNK2 (0.41) MKNK2MKNK1EGFRCYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12036209-B2 Compounds and methods for the targeted degradation of Interleukin-1 receptor-associated kinase 4 polypeptides ARVINAS OPERATIONS, INC. (US) 2024-07-16 US disclosed
WO-2022272060-A1 EP2 ANTAGONIST COMPOUNDS RESERVOIR NEUROSCIENCE, INC. (US) 2022-12-29 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12036209-B2 Compounds and methods for the targeted degradation of Interleukin-1 receptor-associated kinase 4 polypeptides IRAK1, IRAK4, IRAK2 MKNK2 168/4885MKNK1 102/4885EGFR 349/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.