SCHEMBL24833739

SCHEMBL24833739

CC(C)c1ccc(C(=O)N[C@@H]2CCC(=O)NC2=O)nc1

nearest known ligand 0.62

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CRBN Q96SW2 20/20 0.62
DDB1 Q16531 5/20 0.53
IKZF3 Q9UKT9 1/20 0.53
BRD4 O60885 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23485053 1.00 CRBN (0.62) CRBNDDB1IKZF3BRD4
SCHEMBL24833741 1.00 CRBN (0.62) CRBNDDB1IKZF3BRD4
SCHEMBL23594560 0.91 CRBN (0.60) CRBNDDB1IKZF3BRD4
SCHEMBL25626935 0.84 CRBN (0.53) CRBNDDB1IKZF3BRD4
SCHEMBL25627049 0.84 CRBN (0.53) CRBNDDB1IKZF3BRD4
SCHEMBL20128680 0.84 CRBN (0.66) CRBNDDB1IKZF3BRD4
SCHEMBL24890982 0.84 CRBN (0.66) CRBNDDB1IKZF3BRD4
SCHEMBL24316095 0.84 CRBN (0.57) CRBNDDB1IKZF3BRD4
SCHEMBL23594198 0.82 CRBN (0.57) CRBNDDB1IKZF3BRD4
SCHEMBL21946768 0.82 CRBN (0.63) CRBNDDB1IKZF3BRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023093845-A1 CHIMERIC COMPOUND FOR TARGETED DEGRADATION OF ANDROGEN RECEPTOR PROTEIN, PREPARATION METHOD THEREFOR, AND MEDICAL USE THEREOF 江苏恒瑞医药股份有限公司 2023-06-01 WO disclosed
WO-2023274390-A1 BRUTON'S TYROSINE KINASE AND MUTANT DEGRADER, COMPOSITION AND APPLICATION THEREOF 杭州和正医药有限公司 2023-01-05 WO disclosed