SCHEMBL24837469

SCHEMBL24837469

C[C@@H]1CCCCCN1c1nc(Cl)nc2c1CN(C(=O)OC(C)(C)C)C2

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MTOR P42345 2/20 0.39
HPGD P15428 1/20 0.38
EPHX1 P07099 1/20 0.37
ALDH1A1 P00352 3/20 0.34
SMN1; SMN2 Q16637 2/20 0.34
GAA P10253 1/20 0.34
MEN1 O00255 3/20 0.34
KMT2A Q03164 3/20 0.34
MAPT P10636 2/20 0.34
OPRM1 P35372 2/20 0.33
OPRD1 P41143 2/20 0.33
OGFRL1 Q5TC84 2/20 0.33
ALOX5 P09917 1/20 0.33
PARP1 P09874 1/20 0.33
TNKS2 Q9H2K2 1/20 0.33
PARP2 Q9UGN5 1/20 0.33
ATM Q13315 1/20 0.33
RXFP1 Q9HBX9 1/20 0.33
ABL1 P00519 1/20 0.33
RIN1 Q13671 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27191286 1.00 MTOR (0.39) MTORHPGDEPHX1ALDH1A1SMN1; SMN2
SCHEMBL30118094 1.00 MTOR (0.39) MTORHPGDEPHX1ALDH1A1SMN1; SMN2
SCHEMBL29182037 1.00 MTOR (0.39) MTORHPGDEPHX1ALDH1A1SMN1; SMN2
SCHEMBL444134 0.83 MTOR (0.55) MTORPIK3R1PIK3CA
SCHEMBL444716 0.83 MTOR (0.55) MTORPIK3R1PIK3CA
SCHEMBL412835 0.83 MTOR (0.55) MTORPIK3R1PIK3CA
SCHEMBL25265824 0.83 MTOR (0.38) MTORHPGDALDH1A1MEN1KMT2A
SCHEMBL25196466 0.83 MTOR (0.38) MTORHPGDALDH1A1MEN1KMT2A
SCHEMBL20589400 0.83 MTOR (0.38) MTORHPGDALDH1A1MEN1KMT2A
SCHEMBL19358215 0.82 MTOR (0.46) MTORHPGDSMN1; SMN2MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117769554-A Small molecule inhibitors of KRAS muteins 大鹏药品工业株式会社 2024-03-26 CN disclosed
WO-2022250170-A9 SMALL MOLECULE INHIBITORS OF KRAS MUTATED PROTEINS TAIHO PHARMACEUTICAL CO., LTD. (JP) 2023-01-05 WO disclosed