SCHEMBL24845818

SCHEMBL24845818

COC(=O)c1cccc2nc(NC(=O)c3cccc(C(=O)O)c3)n(CCCCCN)c12

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRK1 P41145 2/20 0.47
EHMT2 Q96KQ7 2/20 0.46
MAP3K7 O43318 1/20 0.46
ITK Q08881 2/20 0.45
EHMT1 Q9H9B1 1/20 0.44
KDM4E B2RXH2 3/20 0.44
MEN1 O00255 2/20 0.44
TSHR P16473 2/20 0.44
KMT2A Q03164 2/20 0.44
NPSR1 Q6W5P4 2/20 0.44
USP2 O75604 1/20 0.44
LMNA P02545 1/20 0.44
TP53 P04637 1/20 0.44
HSD17B10 Q99714 1/20 0.44
IRAK4 Q9NWZ3 8/20 0.44
CLK2 P49760 2/20 0.42
CLK4 Q9HAZ1 2/20 0.42
CDK9 P50750 1/20 0.42
MST1R Q04912 1/20 0.42
ADORA2A P29274 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30163798 0.92 EHMT2 (0.48) OPRK1EHMT2MAP3K7ITKEHMT1
SCHEMBL29154814 0.92 EHMT2 (0.48) OPRK1EHMT2MAP3K7ITKEHMT1
SCHEMBL30163779 0.87 STING1 (0.48) OPRK1EHMT2MAP3K7ITKIRAK4
SCHEMBL30163703 0.84 EHMT2 (0.57) OPRK1EHMT2MAP3K7ITKEHMT1
SCHEMBL24845827 0.84 EHMT2 (0.57) OPRK1EHMT2MAP3K7ITKEHMT1
Hydrochloric Acid SCHEMBL30163808 0.83 EHMT2 (0.56) OPRK1EHMT2MAP3K7ITKEHMT1
SCHEMBL24845161 0.82 MAP3K7 (0.41) OPRK1EHMT2MAP3K7ITKEHMT1
SCHEMBL30163826 0.82 MAP3K7 (0.41) OPRK1EHMT2MAP3K7ITKEHMT1
SCHEMBL24845520 0.82 MAP3K7 (0.64) OPRK1EHMT2MAP3K7ITKEHMT1
SCHEMBL24845491 0.82 MAP3K7 (0.64) OPRK1EHMT2MAP3K7ITKEHMT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023275199-A1 MACROCYCLIC TAK1 INHIBITORS AQILION AB (SE) 2023-01-05 WO disclosed