SCHEMBL2485783

SCHEMBL2485783

Cc1ccc2cc(-c3ccc(OCc4c(-c5c(Cl)cccc5Cl)noc4C(C)C)cc3Cl)ccc2c1C(=O)O

nearest known ligand 0.69

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 20/20 0.69
CYP1A2 P05177 2/20 0.66
CYP2C9 P11712 2/20 0.66
NR1I2 O75469 1/20 0.66
CYP3A4 P08684 1/20 0.66
VDR P11473 2/20 0.62
LIFR P42702 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2116096 0.88 NR1H4 (0.85) NR1H4CYP1A2CYP2C9NR1I2CYP3A4
SCHEMBL2112374 0.84 NR1H4 (0.72) NR1H4CYP1A2CYP2C9NR1I2CYP3A4
SCHEMBL2082063 0.82 NR1H4 (0.68) NR1H4CYP1A2CYP2C9NR1I2CYP3A4
SCHEMBL2001397 0.81 NR1H4 (1.00) NR1H4CYP1A2CYP2C9VDR
SCHEMBL2085609 0.81 NR1H4 (0.67) NR1H4CYP1A2CYP2C9NR1I2CYP3A4
SCHEMBL2084444 0.81 NR1H4 (0.65) NR1H4CYP1A2CYP2C9NR1I2CYP3A4
SCHEMBL1179491 0.80 NR1H4 (1.00) NR1H4CYP1A2CYP2C9NR1I2CYP3A4
SCHEMBL16456812 0.80 NR1H4 (0.82) NR1H4CYP1A2CYP2C9NR1I2CYP3A4
SCHEMBL2083720 0.80 NR1H4 (0.73) NR1H4CYP1A2CYP2C9NR1I2CYP3A4
SCHEMBL1179324 0.80 NR1H4 (0.81) NR1H4CYP1A2CYP2C9NR1I2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1962838-B1 FARNESOID X RECEPTOR AGONISTS GLAXOSMITHKLINE LLC (US) 2011-09-28 EP disclosed