SCHEMBL2486972

SCHEMBL2486972

CCCOc1ccc(C)nc1C(=O)N1CCCCC1Cc1cn2ccc(C)c(C)c2n1

nearest known ligand 0.43

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
HCRTR2 O43614 14/20 0.43
HCRTR1 O43613 13/20 0.43
TP53 P04637 1/20 0.39
REN P00797 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2511884 1.00 HCRTR2 (0.43) HCRTR2HCRTR1TP53REN
Hydrochloric Acid SCHEMBL2512239 0.99 HCRTR2 (0.42) HCRTR2HCRTR1TP53REN
SCHEMBL2513353 0.94 HCRTR1 (0.45) HCRTR2HCRTR1
Hydrochloric Acid SCHEMBL2533566 0.93 HCRTR1 (0.44) HCRTR2HCRTR1
SCHEMBL2509592 0.91 HCRTR2 (0.42) HCRTR2HCRTR1
SCHEMBL2486761 0.90 HSD17B10 (0.44) HCRTR2HCRTR1TP53REN
SCHEMBL2515332 0.90 HSD17B10 (0.44) HCRTR2HCRTR1TP53REN
Hydrochloric Acid SCHEMBL2536527 0.90 HCRTR2 (0.42) HCRTR2HCRTR1
SCHEMBL2534343 0.90 HCRTR2 (0.41) HCRTR2HCRTR1
SCHEMBL2510992 0.87 HCRTR1 (0.42) HCRTR2HCRTR1TP53REN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2379550-A1 PIPERIDINE DERIVATIVES USEFUL AS OREXIN ANTAGONISTS Glaxo Group Limited (GB) 2011-10-26 EP claimed
WO-2010072722-A1 PIPERIDINE DERIVATIVES USEFUL AS OREXIN ANTAGONISTS GLAXO GROUP LIMITED (GB) 2010-07-01 WO claimed
EP-2379550-A1 PIPERIDINE DERIVATIVES USEFUL AS OREXIN ANTAGONISTS Glaxo Group Limited (GB) 2011-10-26 EP disclosed
WO-2010072722-A1 PIPERIDINE DERIVATIVES USEFUL AS OREXIN ANTAGONISTS GLAXO GROUP LIMITED (GB) 2010-07-01 WO disclosed