SCHEMBL2487155

SCHEMBL2487155

C#C[C@H](C)N1C(=O)C(C)(C)c2cc3nc(N)[nH]c3cc21

nearest known ligand 0.38

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
FABP6 P51161 1/20 0.38
AURKA O14965 1/20 0.35
AURKB Q96GD4 1/20 0.35
ALDH1A1 P00352 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
TYMS P04818 2/20 0.32
PLAU P00749 1/20 0.31
HTR3E A5X5Y0 1/20 0.31
HTR3B O95264 1/20 0.31
HTR3A P46098 1/20 0.31
BACE1 P56817 1/20 0.31
HTR3D Q70Z44 1/20 0.31
HTR3C Q8WXA8 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3426557 1.00 FABP6 (0.38) FABP6AURKAAURKBALDH1A1TDP1
SCHEMBL2491924 0.79 AURKA (0.45) FABP6AURKAAURKBALDH1A1TDP1
SCHEMBL2490723 0.79 MPI (0.30) TDP1
SCHEMBL13341629 0.76 NPC1 (0.46)
SCHEMBL13367949 0.74 AURKA (0.47) FABP6AURKAAURKBALDH1A1TDP1
SCHEMBL2492686 0.74 AURKA (0.44) FABP6AURKAAURKBALDH1A1TDP1
SCHEMBL3424973 0.73 AURKA (0.44) FABP6AURKAAURKBALDH1A1TDP1
SCHEMBL2491051 0.72 AURKA (0.41) FABP6AURKAAURKBALDH1A1TDP1
SCHEMBL2487407 0.71 AURKA (0.64) FABP6AURKAAURKBALDH1A1TDP1
SCHEMBL2488374 0.71 TDP1 (0.51) ALDH1A1TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1756112-B1 PYRROLOBENZIMIDAZOLONES AND THEIR USE AS ANTIPROLIFERATIVE AGENTS BOEHRINGER INGELHEIM INT (DE) 2011-10-26 EP disclosed