SCHEMBL24879183

SCHEMBL24879183

N[C@@H]1c2ccccc2CC12CCN(c1cnc(Sc3ccc4ncn(Cc5ccccc5)c(=O)c4c3Cl)cn1)CC2

nearest known ligand 0.54

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PTPN11 Q06124 20/20 0.54
MAPK3 P27361 2/20 0.51
MAPK1 P28482 2/20 0.51
KCNH2 Q12809 5/20 0.49
CDK4 P11802 3/20 0.44
CCND3 P30281 3/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30111133 1.00 PTPN11 (0.54) PTPN11MAPK3MAPK1KCNH2CDK4
SCHEMBL24878906 1.00 PTPN11 (0.54) PTPN11MAPK3MAPK1KCNH2CDK4
SCHEMBL24878748 0.91 PTPN11 (0.62) PTPN11MAPK3MAPK1KCNH2
SCHEMBL30110972 0.91 PTPN11 (0.62) PTPN11MAPK3MAPK1KCNH2
SCHEMBL24878872 0.91 PTPN11 (0.62) PTPN11MAPK3MAPK1KCNH2
SCHEMBL24879124 0.91 PTPN11 (0.62) PTPN11MAPK3MAPK1KCNH2
SCHEMBL30111268 0.91 PTPN11 (0.62) PTPN11MAPK3MAPK1KCNH2
SCHEMBL30987334 0.89 PTPN11 (0.53) PTPN11MAPK3MAPK1KCNH2CDK4
SCHEMBL24879085 0.89 PTPN11 (0.54) PTPN11MAPK3MAPK1KCNH2CDK4
SCHEMBL30111100 0.89 PTPN11 (0.54) PTPN11MAPK3MAPK1KCNH2CDK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12029739-B2 SHP2 inhibitor and use thereof KANAPH THERAPEUTICS INC. (KR) 2024-07-09 US disclosed
US-12029739-B2 SHP2 inhibitor and use thereof KANAPH THERAPEUTICS INC. (KR) 2024-07-09 US disclosed
US-12029739-B2 SHP2 inhibitor and use thereof KANAPH THERAPEUTICS INC. (KR) 2024-07-09 US disclosed
CN-117916242-A SHP2 inhibitors and uses thereof 治纳辅医药科技有限公司 2024-04-19 CN disclosed
WO-2023282702-A1 SHP2 INHIBITOR AND USE THEREOF 주식회사 카나프테라퓨틱스 2023-01-12 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12029739-B2 SHP2 inhibitor and use thereof PTPN1, PTPN5, PTPN2 PTPN11 16/4885MAPK3 389/4885MAPK1 272/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.