SCHEMBL2490826

SCHEMBL2490826

CCS(=O)(=O)C1(c2cc(N3CCOCC3C)nc(Cl)n2)CCN(C(=O)O)CC1

nearest known ligand 0.45

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ATR Q13535 20/20 0.45
ATRIP Q8WXE1 4/20 0.45
MTOR P42345 5/20 0.42
TAF1 P21675 3/20 0.42
PRKDC P78527 2/20 0.42
KCNH2 Q12809 4/20 0.42
PIK3CA P42336 3/20 0.42
PIK3R1 P27986 1/20 0.42
ATM Q13315 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4203309 0.91 ATR (0.54) ATRATRIPMTORTAF1PRKDC
SCHEMBL2489919 0.90 ATR (0.52) ATRATRIPMTORTAF1PRKDC
SCHEMBL6518645 0.90 ATR (0.52) ATRATRIPMTORTAF1PRKDC
SCHEMBL4202234 0.90 ATR (0.52) ATRATRIPMTORTAF1PRKDC
SCHEMBL2492774 0.89 PIK3R1 (0.44) ATRATRIPMTORTAF1PRKDC
SCHEMBL6524143 0.89 PIK3R1 (0.44) ATRATRIPMTORTAF1PRKDC
SCHEMBL4197531 0.88 ATR (0.49) ATRATRIPMTORTAF1PRKDC
SCHEMBL2489905 0.88 ATR (0.49) ATRATRIPMTORTAF1PRKDC
SCHEMBL2489908 0.88 ATR (0.49) ATRATRIPMTORTAF1PRKDC
SCHEMBL2490413 0.88 MTOR (0.50) ATRATRIPMTORTAF1PRKDC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2379530-A1 PYRIMIDINE INDOLE DERIVATIVES FOR TREATING CANCER AstraZeneca AB (SE) 2011-10-26 EP disclosed
WO-2010073034-A1 PYRIMIDINE INDOLE DERIVATIVES FOR TREATING CANCER ASTRAZENECA AB (SE) 2010-07-01 WO disclosed