SCHEMBL24920918

SCHEMBL24920918

Cc1ccc(C2(c3ccc(OCc4ccnc(-c5ncc[nH]5)n4)cc3)CCC2)cc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX5AP P20292 6/20 0.38
NISCH Q9Y2I1 1/20 0.36
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34
CYP19A1 P11511 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
SMO Q99835 2/20 0.34
MAPK14 Q16539 1/20 0.34
NPC1 O15118 4/20 0.34
RAB9A P51151 4/20 0.34
SMN1; SMN2 Q16637 4/20 0.34
PDE10A Q9Y233 1/20 0.34
HPGD P15428 1/20 0.33
KDM4E B2RXH2 1/20 0.32
NFKB1 P19838 1/20 0.32
HTT P42858 1/20 0.32
NFKB2 Q00653 1/20 0.32
RELA Q04206 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24920739 0.89 NISCH (0.36) ALOX5APNISCHCYP1A2CYP3A4CYP2D6
SCHEMBL24920920 0.83 NPC1 (0.36) ALOX5APNPC1RAB9ASMN1; SMN2PDE10A
SCHEMBL24921215 0.81 NPC1 (0.40) ALOX5APCYP19A1NPC1RAB9ASMN1; SMN2
SCHEMBL24920850 0.81 ALOX5AP (0.35) ALOX5APCYP19A1NPC1RAB9ASMN1; SMN2
SCHEMBL24921642 0.81 NISCH (0.40) NISCHCYP1A2CYP3A4CYP2D6CYP19A1
SCHEMBL24920875 0.80 ALOX5AP (0.35) ALOX5APNPC1RAB9ASMN1; SMN2PDE10A
SCHEMBL24920884 0.80 ALOX5AP (0.35) ALOX5APNPC1RAB9ASMN1; SMN2HPGD
SCHEMBL24920877 0.79 NPC1 (0.35) ALOX5APCYP1A2CYP2D6CYP19A1CYP2C9
SCHEMBL24920909 0.79 NPC1 (0.38) ALOX5APCYP19A1NPC1RAB9ASMN1; SMN2
SCHEMBL24921252 0.78 NPC1 (0.39) ALOX5APNPC1RAB9ASMN1; SMN2PDE10A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023006097-A1 BIFUNCTIONAL CHIMERIC HETEROCYCLIC COMPOUND AND USE THEREOF AS ANDROGEN RECEPTOR DEGRADER 海创药业股份有限公司 2023-02-02 WO disclosed