SCHEMBL24923036

SCHEMBL24923036

BOC(=O)CN1CCNCCNCc2cccc(n2)C1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CXCR4 P61073 7/20 0.51
ADRB1 P08588 1/20 0.34
KDM4E B2RXH2 2/20 0.33
ALDH1A1 P00352 1/20 0.33
JAK3 P52333 1/20 0.32
HTR2A P28223 2/20 0.32
HTR2C P28335 1/20 0.32
SLC6A4 P31645 1/20 0.32
HSD17B10 Q99714 2/20 0.31
HTR3E A5X5Y0 1/20 0.31
HTR3B O95264 1/20 0.31
CYP1A2 P05177 1/20 0.31
HTR1A P08908 1/20 0.31
CYP2D6 P10635 1/20 0.31
NCF1 P14598 1/20 0.31
TSHR P16473 1/20 0.31
NFKB1 P19838 1/20 0.31
HTR1D P28221 1/20 0.31
HTR1B P28222 1/20 0.31
HTR7 P34969 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19058527 0.89 CXCR4 (0.50) CXCR4ADRB1ALDH1A1HSD17B10
SCHEMBL21427272 0.86 CXCR4 (0.55) CXCR4ADRB1KDM4EALDH1A1SIGMAR1
SCHEMBL12342819 0.80 MEN1 (0.44) CXCR4ADRB1KDM4EALDH1A1HTR2C
SCHEMBL12629018 0.79 KMT2A (0.44) CXCR4ADRB1KDM4EALDH1A1HTR2A
SCHEMBL9213719 0.79 CXCR4 (0.49) CXCR4ADRB1KDM4EALDH1A1HTR2A
SCHEMBL21427211 0.77 CXCR4 (0.52) CXCR4ADRB1KDM4EALDH1A1
SCHEMBL24922952 0.77 HTR2A (0.33) KDM4EALDH1A1HTR2AHTR2CSLC6A4
SCHEMBL4359497 0.76 MEN1 (0.41) CXCR4ALDH1A1TSHR
SCHEMBL21906528 0.76 CXCR4 (0.61) CXCR4ADRB1JAK3SIGMAR1
SCHEMBL674043 0.75 CXCR4 (0.83) CXCR4SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023006938-A1 MACROCYCLIC LIGANDS WITH PICOLINATE GROUP(S), COMPLEXES AND MEDICAL USES THEREOF GUERBET (FR) 2023-02-02 WO disclosed
EP-4124361-A1 MACROCYCLIC LIGANDS WITH PICOLINATE GROUP(S), COMPLEXES THEREOF AND MEDICAL USES THEREOF Guerbet (FR) 2023-02-01 EP disclosed