SCHEMBL24973

SCHEMBL24973

CSCCCNC(=O)c1ccc2c(c1)NC(=O)C2

nearest known ligand 0.58

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SMYD3 Q9H7B4 8/20 0.58
HDAC3 O15379 3/20 0.57
HDAC1 Q13547 3/20 0.57
CRBN Q96SW2 2/20 0.51
HDAC6 Q9UBN7 3/20 0.50
PDGFRA P16234 2/20 0.50
HDAC4 P56524 2/20 0.50
HDAC2 Q92769 2/20 0.50
HDAC8 Q9BY41 2/20 0.50
HDAC9 Q9UKV0 2/20 0.50
EPHX2 P34913 1/20 0.49
NAMPT P43490 1/20 0.48
PDGFRB P09619 1/20 0.48
KDR P35968 1/20 0.48
TP53 P04637 1/20 0.46
HPGD P15428 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26301 0.91 SMYD3 (0.71) SMYD3HDAC3HDAC1HDAC6PDGFRA
SCHEMBL29528307 0.81 SMYD3 (0.59) SMYD3HDAC3HDAC1CRBNHDAC6
SCHEMBL23175705 0.78 HDAC2 (0.58) SMYD3HDAC3HDAC1CRBNHDAC6
SCHEMBL5316057 0.76 CRBN (0.81) SMYD3HDAC3HDAC1CRBNHDAC6
SCHEMBL4935353 0.76 SMYD3 (0.74) SMYD3HDAC3HDAC1HDAC6HDAC4
SCHEMBL29899620 0.75 SMYD3 (0.54) SMYD3
SCHEMBL23143521 0.75 SMYD3 (0.54) SMYD3
SCHEMBL3207365 0.75 SMYD3 (0.72) SMYD3HDAC3HDAC1HDAC6HDAC4
SCHEMBL18006544 0.74 EPHX2 (0.54) SMYD3HDAC3HDAC1CRBNHDAC6
SCHEMBL3182105 0.74 SMYD3 (0.71) SMYD3HDAC3HDAC1HDAC6HDAC4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012025726-A1 Novel Hybrid Compounds UNIVERSITY OF GREENWICH (GB) 2012-03-01 WO disclosed
WO-2012025726-A1 Novel Hybrid Compounds UNIVERSITY OF GREENWICH (GB) 2012-03-01 WO disclosed