SCHEMBL24975338

SCHEMBL24975338

CN(C[C@H]1Cc2c(cccc2N2CCN3CCOC[C@H]3C2)CN1)C1CCCc2cccnc21

nearest known ligand 0.86

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CXCR4 P61073 20/20 0.86
CHRM2 P08172 7/20 0.82
CHRM4 P08173 7/20 0.82
CHRM5 P08912 7/20 0.82
CHRM1 P11229 7/20 0.82
CHRM3 P20309 7/20 0.82
CYP2D6 P10635 9/20 0.80
CYP3A4 P08684 4/20 0.80
KCNH2 Q12809 1/20 0.70
CYP2C9 P11712 1/20 0.69

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21744280 1.00 CXCR4 (0.86) CXCR4CHRM2CHRM4CHRM5CHRM1
SCHEMBL30239406 1.00 CXCR4 (0.86) CXCR4CHRM2CHRM4CHRM5CHRM1
SCHEMBL21744626 1.00 CXCR4 (0.86) CXCR4CHRM2CHRM4CHRM5CHRM1
SCHEMBL21744358 0.93 CXCR4 (0.80) CXCR4CHRM2CHRM4CHRM5CHRM1
SCHEMBL21744261 0.93 CXCR4 (0.80) CXCR4CHRM2CHRM4CHRM5CHRM1
SCHEMBL21744415 0.93 CXCR4 (1.00) CXCR4CHRM2CHRM4CHRM5CHRM1
SCHEMBL21744281 0.93 CXCR4 (1.00) CXCR4CHRM2CHRM4CHRM5CHRM1
SCHEMBL21744235 0.90 CXCR4 (1.00) CXCR4CHRM2CHRM4CHRM5CHRM1
SCHEMBL21744749 0.90 CXCR4 (1.00) CXCR4CHRM2CHRM4CHRM5CHRM1
SCHEMBL21744236 0.90 CXCR4 (1.00) CXCR4CHRM2CHRM4CHRM5CHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023003862-A1 CXCR4 MODULATORS AND USES RELATED THERETO EMORY UNIVERSITY (US) 2023-01-26 WO disclosed