SCHEMBL24975800

SCHEMBL24975800

Cc1cc(-c2ccccc2C(=O)OC(C)(C)C)c2cc(C(=O)N3CCOCC3)ccc2n1

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.46
PKM P14618 1/20 0.46
HPGD P15428 3/20 0.43
USP2 O75604 1/20 0.41
ALDH1A1 P00352 1/20 0.41
TP53 P04637 1/20 0.41
POLB P06746 1/20 0.41
TSHR P16473 1/20 0.41
HSD17B10 Q99714 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2C9 P11712 1/20 0.41
PDE4B Q07343 1/20 0.41
HSP90AA1 P07900 1/20 0.41
HSP90AB1 P08238 1/20 0.41
PDCD1 Q15116 1/20 0.41
CD274 Q9NZQ7 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31428793 1.00 KDM4E (0.46) KDM4EPKMHPGDUSP2ALDH1A1
SCHEMBL31428482 0.89 HPGD (0.41) HPGDALDH1A1TSHRCYP1A2CYP3A4
SCHEMBL24975789 0.89 HPGD (0.41) HPGDALDH1A1TSHRCYP1A2CYP3A4
SCHEMBL31428610 0.86 GRM2 (0.46) KDM4EPKMHPGDUSP2ALDH1A1
SCHEMBL31428552 0.85 MEN1 (0.46) KDM4EPKMHPGDTSHRPDCD1
SCHEMBL31428537 0.83 PDCD1 (0.52) KDM4EPKMHPGDUSP2ALDH1A1
SCHEMBL31428699 0.82 HTR2C (0.53) KDM4EPKMHPGDUSP2ALDH1A1
SCHEMBL31428513 0.81 PDCD1 (0.53) KDM4EPKMHPGDUSP2ALDH1A1
SCHEMBL24977037 0.79 CNR2 (0.47) ALDH1A1
SCHEMBL31428639 0.79 CNR2 (0.47) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023008577-A1 RAS/RAF BINDING INHIBITOR COMPOUND 国立大学法人神戸大学 2023-02-02 WO disclosed