SCHEMBL2498233

SCHEMBL2498233

CC(C(=O)O)N1CCN(Cc2ccc3ncc(-c4cc(O[C@H](C)c5ccccc5Cl)c(C(N)=O)s4)n3c2)CC1

nearest known ligand 0.74

Predicted protein targets (top 1)

geneUniProtsupporting neighboursconfidence
PLK1 P53350 20/20 0.74

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4579608 0.92 PLK1 (0.76) PLK1
SCHEMBL2523836 0.92 PLK1 (0.78) PLK1
SCHEMBL2516478 0.92 PLK1 (0.80) PLK1
SCHEMBL2521826 0.91 PLK1 (0.79) PLK1
SCHEMBL2523908 0.90 PLK1 (0.76) PLK1
SCHEMBL2518635 0.90 PLK1 (0.76) PLK1
SCHEMBL2526052 0.90 PLK1 (0.78) PLK1
SCHEMBL2518636 0.90 PLK1 (0.76) PLK1
SCHEMBL2526050 0.90 PLK1 (0.78) PLK1
SCHEMBL2523899 0.90 PLK1 (0.76) PLK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8030327-B2 3-[1-(2-chlorophenyl)ethoxy]-5-imidazo[1,2-a]pyridin-3-ylthiophene-2-carboxyamide; polo like kinase inhibitor; antitumor and anticarcinogenic agent; mitotic phase (M phase) of the cell cycle MDS K.K. (JP) 2011-10-04 US disclosed