SCHEMBL2500287

SCHEMBL2500287

OC1CCCCC1n1ccc2cc(-c3ccn4c(CC(F)(F)F)cnc4c3Cl)ccc21

nearest known ligand 0.78

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
GRM2 Q14416 20/20 0.78
GRM7 Q14831 1/20 0.78

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL565532 0.88 GRM2 (1.00) GRM2GRM7
SCHEMBL565531 0.88 GRM2 (1.00) GRM2GRM7
SCHEMBL564687 0.83 GRM2 (0.79) GRM2GRM7
SCHEMBL564686 0.83 GRM2 (0.79) GRM2GRM7
SCHEMBL566125 0.77 GRM2 (0.64) GRM2GRM7
SCHEMBL19139297 0.74 GRM2 (0.83) GRM2GRM7
SCHEMBL921517 0.73 GRM2 (1.00) GRM2GRM7
SCHEMBL12907976 0.73 GRM2 (1.00) GRM2GRM7
SCHEMBL565359 0.72 GRM2 (0.79) GRM2GRM7
SCHEMBL565358 0.72 GRM2 (0.79) GRM2GRM7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2373649-A1 INDOLE AND BENZOXAZINE DERIVATIVES AS MODULATORS OF METABOTROPIC GLUTAMATE RECEPTORS Ortho-McNeil-Janssen Pharmaceuticals, Inc. (US) 2011-10-12 EP disclosed
WO-2010060589-A1 INDOLE AND BENZOXAZINE DERIVATIVES AS MODULATORS OF METABOTROPIC GLUTAMATE RECEPTORS ORTHO-MCNEIL-JANSSEN PHARMACEUTICALS, INC. (US) 2010-06-03 WO disclosed