SCHEMBL2500720

SCHEMBL2500720

O=C(Cc1cccc2nc[nH]c12)OC(=O)C(F)(F)F

nearest known ligand 0.32

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.32
HPGD P15428 1/20 0.32
APOBEC3A P31941 1/20 0.32
APOBEC3G Q9HC16 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2498738 0.83 PARP1 (0.34) PARP1
Trifluoroacetic Acid SCHEMBL2500718 0.80 GRIN2D (0.41) PARP1
SCHEMBL2495511 0.80 CDK2 (0.33) PARP1HPGD
SCHEMBL2500031 0.76 GRIN2D (0.47) PARP1
Acetic Acid SCHEMBL2498732 0.72 GRIN2D (0.44) PARP1
SCHEMBL2496167 0.69 CYP4F2 (0.33) PARP1HPGD
SCHEMBL2501354 0.69 PARP1 (0.40) PARP1
SCHEMBL7346990 0.69 PARP1 (0.43) PARP1
SCHEMBL27457721 0.69 PARP1 (0.40) PARP1HPGD
SCHEMBL14755023 0.69 KCNJ5 (0.47) HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2373628-A1 NOVEL COMPOUNDS Glaxo Group Limited (GB) 2011-10-12 EP disclosed
WO-2010070021-A1 NOVEL COMPOUNDS GLAXO GROUP LIMITED (GB) 2010-06-24 WO disclosed