SCHEMBL25019142

SCHEMBL25019142

C[C@H]1CCN2C(=O)c3c(O)c(=O)c(C(=O)NCc4ccc(F)cc4)cn3CC2(C)N1C

nearest known ligand 0.54

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
SLC22A2 O15244 6/20 0.46
CYP3A4 P08684 1/20 0.46
TMEM97 Q5BJF2 1/20 0.46
ABCG2 Q9UNQ0 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10283767 0.96 SLC22A2 (0.45) SLC22A2CYP3A4TMEM97ABCG2
SCHEMBL19178164 0.90 SLC22A2 (0.46) SLC22A2CYP3A4TMEM97ABCG2
SCHEMBL23615832 0.89 SLC22A2 (0.45) SLC22A2CYP3A4TMEM97ABCG2
SCHEMBL20008022 0.87 SLC22A2 (0.44) SLC22A2CYP3A4TMEM97ABCG2
SCHEMBL23615880 0.85 SLC22A2 (0.44) SLC22A2CYP3A4TMEM97ABCG2
SCHEMBL19177060 0.81 SLC22A2 (0.42) SLC22A2CYP3A4TMEM97ABCG2
SCHEMBL19177883 0.79 TP53 (0.42)
SCHEMBL18462047 0.79 SLC22A2 (0.45) SLC22A2CYP3A4TMEM97ABCG2
SCHEMBL19071817 0.79 SLC22A2 (0.57) SLC22A2CYP3A4TMEM97ABCG2
SCHEMBL81635 0.79 SLC22A2 (0.57) SLC22A2CYP3A4TMEM97ABCG2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3045206-B2 POLYCYCLIC CARBAMOYLPYRIDONE DERIVATIVE HAVING HIV INTEGRASE INHIBITORY ACTIVITY VIIV HEALTHCARE CO (US) 2023-02-15 EP disclosed