SCHEMBL25035630

SCHEMBL25035630

CC(C)n1c(=O)c(-c2cc(F)c(NS(=O)(=O)C3CCCCC3)c(F)c2)cc2cnc(N)nc21

nearest known ligand 0.39

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALOX5AP P20292 4/20 0.39
FEN1 P39748 3/20 0.39
ERN1 O75460 4/20 0.38
FGFR1 P11362 1/20 0.37
FGFR2 P21802 1/20 0.37
FGFR4 P22455 1/20 0.37
FGFR3 P22607 1/20 0.37
BRAF P15056 1/20 0.37
PIK3CA P42336 7/20 0.36
MTOR P42345 3/20 0.36
ABL1 P00519 1/20 0.33
ELANE P08246 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25035653 0.89 ERN1 (0.47) ALOX5APFEN1ERN1BRAFPIK3CA
SCHEMBL25035487 0.88 ERN1 (0.47) ALOX5APFEN1ERN1BRAFPIK3CA
SCHEMBL25035632 0.82 ERN1 (0.59) ERN1FGFR1
SCHEMBL25035337 0.79 BRAF (0.44) ALOX5APFEN1ERN1FGFR1FGFR2
SCHEMBL25035529 0.78 ERN1 (0.50) ALOX5APFEN1ERN1BRAFPIK3CA
SCHEMBL25035330 0.78 ERN1 (0.46) ALOX5APFEN1ERN1FGFR1FGFR2
SCHEMBL25034120 0.78 ERN1 (0.52) ERN1FGFR1FGFR2FGFR4FGFR3
SCHEMBL25035269 0.78 ERN1 (0.45) ERN1FGFR1FGFR2FGFR4FGFR3
SCHEMBL25035327 0.78 ERN1 (0.46) ERN1FGFR1FGFR2FGFR4FGFR3
SCHEMBL25034117 0.77 ERN1 (0.46) ERN1FGFR1FGFR2FGFR4FGFR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230047209-A1 PYRIDO-PYRIMIDINONE AND PTERIDINONE COMPOUNDS AND METHODS OF USE PARAZA PHARMA, INC. (CA) 2023-02-16 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230047209-A1 PYRIDO-PYRIMIDINONE AND PTERIDINONE COMPOUNDS AND METHODS OF USE TYMP, TYMS, DPYD ALOX5AP 1186/4885FEN1 50/4885ERN1 3167/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.