SCHEMBL25042628

SCHEMBL25042628

CC(C)Sc1ccc(-c2cnc(N)c(-c3cc(-c4ccc(N)cc4)no3)n2)cc1

nearest known ligand 0.58

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ATR Q13535 20/20 0.58
ATM Q13315 9/20 0.58
GSK3B P49841 3/20 0.58
PRKDC P78527 4/20 0.56
JAK2 O60674 1/20 0.52
ABL1 P00519 1/20 0.52
KIT P10721 1/20 0.52
SERPINA2 P20848 1/20 0.52
PIK3R1 P27986 1/20 0.52
FLT4 P35916 1/20 0.52
FLT3 P36888 1/20 0.52
PIK3CA P42336 1/20 0.52
MTOR P42345 1/20 0.52
SYK P43405 1/20 0.52
GSK3A P49840 1/20 0.52
MAP3K9 P80192 1/20 0.52
KCNH2 Q12809 1/20 0.52
MERTK Q12866 1/20 0.52
DYRK2 Q92630 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24709136 0.87 ATR (0.71) ATRATMGSK3BPRKDCJAK2
SCHEMBL25042981 0.85 ATR (0.50) ATRATMGSK3BPRKDCJAK2
SCHEMBL25042554 0.85 ATR (0.52) ATRATMGSK3BPRKDCJAK2
SCHEMBL25042558 0.85 ATR (0.59) ATRATMGSK3BPRKDCJAK2
SCHEMBL25042957 0.84 ATR (0.52) ATRATMGSK3BPRKDCJAK2
SCHEMBL25042597 0.84 ATR (0.49) ATRATMGSK3BPRKDCJAK2
SCHEMBL25042606 0.84 ATR (0.49) ATRATMGSK3BPRKDCJAK2
SCHEMBL19672802 0.84 ATR (0.60) ATRATMGSK3BPRKDCJAK2
SCHEMBL25042644 0.84 ATR (0.51) ATRATMGSK3BPRKDCJAK2
SCHEMBL25042544 0.83 ATR (0.56) ATRATMGSK3BPRKDCJAK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023016525-A1 COMPOUND AS ATR KINASE INHIBITOR 苏州爱科百发生物医药技术有限公司 2023-02-16 WO disclosed