SCHEMBL25075271

SCHEMBL25075271

C[C@@H](COc1cc(Cl)ncc1Cl)NC(=O)OC(C)(C)C

nearest known ligand 0.48

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
AAK1 Q2M2I8 8/20 0.48
TRPA1 O75762 1/20 0.43
CNR2 P34972 6/20 0.40
CNR1 P21554 1/20 0.40
STK17B O94768 1/20 0.40
STK17A Q9UEE5 1/20 0.40
IRAK4 Q9NWZ3 1/20 0.38
ACACB O00763 1/20 0.38
PTGER1 P34995 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29169125 1.00 AAK1 (0.48) AAK1TRPA1CNR2CNR1STK17B
SCHEMBL29169087 0.89 AAK1 (0.46) AAK1TRPA1IRAK4ACACBPTGER1
SCHEMBL29168923 0.88 AAK1 (0.47) AAK1TRPA1
SCHEMBL25075435 0.88 AAK1 (0.47) AAK1TRPA1
SCHEMBL25397733 0.81 AAK1 (0.43) AAK1TRPA1
SCHEMBL25397736 0.81 AAK1 (0.43) AAK1TRPA1
SCHEMBL29882519 0.80 AAK1 (0.51) AAK1TRPA1PTGER1
SCHEMBL23609241 0.80 AAK1 (0.51) AAK1TRPA1PTGER1
SCHEMBL28850131 0.80 AAK1 (0.51) AAK1TRPA1PTGER1
SCHEMBL25075354 0.80 AAK1 (0.43) AAK1TRPA1IRAK4ACACB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023020479-A1 PARP7 INHIBITOR AND APPLICATION THEREOF 重庆华森制药股份有限公司 2023-02-23 WO disclosed