SCHEMBL251264

SCHEMBL251264

COc1cc(-c2c(C#N)c(Nc3ccccc3)nc(Sc3ccccc3)c2C#N)ccc1F

nearest known ligand 0.45

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 6/20 0.45
ADORA1 P30542 5/20 0.45
DCUN1D1 Q96GG9 1/20 0.42
MAPT P10636 4/20 0.42
NPSR1 Q6W5P4 1/20 0.42
RXFP1 Q9HBX9 1/20 0.42
ALDH1A1 P00352 1/20 0.40
ADORA2B P29275 2/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
ABCG2 Q9UNQ0 3/20 0.39
PRKCQ Q04759 1/20 0.38
THRB P10828 1/20 0.38
TP53 P04637 1/20 0.37
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3328078 0.84 MAPT (0.60) ADORA2AADORA1MAPTNPSR1RXFP1
SCHEMBL3333404 0.66 MAPT (0.81) ADORA2AADORA1MAPTNPSR1RXFP1
SCHEMBL3339298 0.65 KDM4E (0.51) ADORA2AADORA1MAPTNPSR1RXFP1
SCHEMBL244863 0.64 ADORA1 (0.61) ADORA2AADORA1MAPTNPSR1RXFP1
SCHEMBL245478 0.64 ADORA1 (0.65) ADORA2AADORA1MAPTNPSR1RXFP1
SCHEMBL4031424 0.64 ADORA1 (0.48) ADORA2AADORA1MAPTNPSR1ALDH1A1
SCHEMBL6462984 0.63 MAPT (0.59) ADORA2AADORA1MAPTNPSR1RXFP1
SCHEMBL3548799 0.63 KDM4E (0.49) ADORA2AADORA1MAPTNPSR1RXFP1
SCHEMBL3605617 0.63 PRF1 (0.44) ADORA1MAPTNPSR1RXFP1ALDH1A1
SCHEMBL13879906 0.63 ADORA1 (0.50) ADORA2AADORA1MAPTNPSR1RXFP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2588454-A1 SUBSTITUTED DICYANOPYRIDINES AND USE THEREOF Bayer Intellectual Property GmbH (DE) 2013-05-08 EP disclosed
WO-2012000945-A1 SUBSTITUTED DICYANOPYRIDINES AND USE THEREOF BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2012-01-05 WO disclosed