SCHEMBL2513019

SCHEMBL2513019

Cn1c(NC2[C@H]3CN(C(=O)O)C[C@@H]23)nc(-c2ccncc2)cc1=O

nearest known ligand 0.55

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 20/20 0.55
CYP1A2 P05177 3/20 0.45
CYP2D6 P10635 3/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2513018 1.00 GSK3B (0.55) GSK3BCYP1A2CYP2D6
SCHEMBL2513017 1.00 GSK3B (0.55) GSK3BCYP1A2CYP2D6
SCHEMBL2513016 1.00 GSK3B (0.55) GSK3BCYP1A2CYP2D6
SCHEMBL2488133 0.91 GSK3B (0.53) GSK3BCYP1A2CYP2D6
SCHEMBL2488135 0.91 GSK3B (0.53) GSK3BCYP1A2CYP2D6
SCHEMBL14302424 0.91 GSK3B (0.53) GSK3BCYP1A2CYP2D6
SCHEMBL2488137 0.91 GSK3B (0.53) GSK3BCYP1A2CYP2D6
SCHEMBL2490764 0.89 GSK3B (0.61) GSK3BCYP1A2CYP2D6
SCHEMBL2490762 0.89 GSK3B (0.61) GSK3BCYP1A2CYP2D6
SCHEMBL2490759 0.89 GSK3B (0.61) GSK3BCYP1A2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2057141-B1 PYRIMIDONE COMPOUNDS AS GSK-3 INHIBITORS PFIZER PROD INC (US) 2011-10-26 EP disclosed