SCHEMBL25147666

SCHEMBL25147666

CC(C)(C)OC(=O)N1CCc2ncc(CC(F)(F)F)cc2C1

nearest known ligand 0.49

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.49
NR1H2 P55055 2/20 0.49
ESR2 Q92731 1/20 0.47
HPGDS O60760 2/20 0.41
MAPK1 P28482 1/20 0.39
GPR119 Q8TDV5 1/20 0.38
SLC34A1 Q06495 1/20 0.38
LIPG Q9Y5X9 1/20 0.38
ABHD6 Q9BV23 1/20 0.37
FGFR3 P22607 1/20 0.37
KDR P35968 1/20 0.37
NAMPT P43490 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30332059 1.00 MAPT (0.49) MAPTNR1H2ESR2HPGDSMAPK1
SCHEMBL10313002 0.87 MAPT (0.52) MAPTNR1H2ESR2HPGDSMAPK1
SCHEMBL10313009 0.87 MAPT (0.52) MAPTNR1H2ESR2HPGDSMAPK1
SCHEMBL13226354 0.83 MAPT (0.48) MAPTNR1H2ESR2HPGDSMAPK1
SCHEMBL2211825 0.83 MAPT (0.52) MAPTNR1H2ESR2
SCHEMBL29507818 0.82 NR1H2 (0.64) MAPTNR1H2ESR2HPGDSMAPK1
SCHEMBL3002453 0.82 NR1H2 (0.64) MAPTNR1H2ESR2HPGDSMAPK1
SCHEMBL29421798 0.82 ESR2 (0.47) MAPTNR1H2ESR2GPR119
SCHEMBL13226239 0.81 ESR2 (0.63) MAPTNR1H2ESR2HPGDSMAPK1
SCHEMBL25153126 0.81 MAPT (0.55) MAPTNR1H2ESR2HPGDSMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023064585-A1 7,8-DIHYDRO-5H-1,6-NAPHTHYRIDINE DERIVATIVES AS POSITIVE ALLOSTERIC MODULATORS OF THE MUSCARINIC ACETYLCHOLINE RECEPTOR M4 FOR TREATING NEUROLOGICAL AND PSYCHIATRIC DISORDERS VANDERBILT UNIVERSITY (US) 2023-04-20 WO disclosed