SCHEMBL25190852

SCHEMBL25190852

Cc1nc2cccc(C)c2c(C)c1C(N)=O

nearest known ligand 0.47

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
EPHB4 P54760 3/20 0.44
TP53 P04637 1/20 0.43
HSD17B10 Q99714 1/20 0.43
HTT P42858 2/20 0.42
ELANE P08246 5/20 0.41
PARP1 P09874 1/20 0.41
PDE10A Q9Y233 1/20 0.41
DHODH Q02127 1/20 0.40
ACHE P22303 1/20 0.38
WEE1 P30291 2/20 0.38
PKMYT1 Q99640 2/20 0.38
KDM4E B2RXH2 1/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
EPHB3 P54753 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5304399 0.86 EPHB4 (0.43) EPHB4ELANEPARP1DHODHACHE
SCHEMBL10258857 0.85 PDE10A (0.54) TP53HSD17B10HTTELANEPARP1
SCHEMBL28881597 0.81 DHODH (0.51) EPHB4PDE10ADHODHKDM4EMEN1
SCHEMBL28386669 0.79 ELANE (0.42) EPHB4ELANEPARP1DHODHACHE
SCHEMBL14883918 0.77 HTT (0.69) TP53HSD17B10HTTPDE10ADHODH
SCHEMBL8168011 0.76 PDE10A (0.47) EPHB4TP53HSD17B10HTTPDE10A
SCHEMBL618719 0.76 HSD17B10 (0.53) TP53HSD17B10HTTELANEPARP1
SCHEMBL29041769 0.75 ELANE (0.42) EPHB4ELANEPARP1DHODHACHE
SCHEMBL3885065 0.75 ELANE (0.47) ELANEPARP1ACHE
SCHEMBL29791541 0.75 ELANE (0.47) ELANEPARP1ACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230158156-A1 BIFUNCTIONAL MOLECULES AND METHODS OF USING THEREOF FLAGSHIP PIONEERING, INC. (US) 2023-05-25 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230158156-A1 BIFUNCTIONAL MOLECULES AND METHODS OF USING THEREOF EFTUD2, SNRPE, DDX21 EPHB4 3431/4885TP53 333/4885HSD17B10 3540/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.