SCHEMBL25211008

SCHEMBL25211008

CC(=O)c1ccc2c(c1)[n+]([O-])nc(NCCC(=O)O)[n+]2[O-]

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 3/20 0.38
CA2 P00918 3/20 0.38
CA12 O43570 2/20 0.38
CA9 Q16790 2/20 0.38
POLB P06746 1/20 0.36
KMT2A Q03164 2/20 0.35
KDM4E B2RXH2 2/20 0.35
MEN1 O00255 1/20 0.34
APAF1 O14727 1/20 0.34
HSD17B10 Q99714 3/20 0.33
HPGD P15428 4/20 0.32
GCGR P47871 1/20 0.32
L3MBTL1 Q9Y468 2/20 0.31
TDP1 Q9NUW8 1/20 0.31
ALDH1A1 P00352 3/20 0.30
MAPT P10636 3/20 0.30
APEX1 P27695 1/20 0.30
AKR1C3 P42330 1/20 0.30
AKR1C2 P52895 1/20 0.30
AKR1C1 Q04828 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29864943 1.00 CA1 (0.38) CA1CA2CA12CA9POLB
SCHEMBL25210832 0.85 HTT (0.35) CA1CA2CA12CA9KMT2A
SCHEMBL29864546 0.85 HTT (0.35) CA1CA2CA12CA9KMT2A
SCHEMBL29864507 0.83 CA12 (0.40) CA1CA2CA12CA9POLB
SCHEMBL25074666 0.83 APEX1 (0.45) CA1CA2CA12CA9KMT2A
SCHEMBL29864646 0.83 APEX1 (0.45) CA1CA2CA12CA9KMT2A
SCHEMBL25074972 0.83 CA12 (0.40) CA1CA2CA12CA9POLB
SCHEMBL25211012 0.82 TDP1 (0.48) CA1CA2CA12CA9POLB
SCHEMBL25210259 0.78 TDP1 (0.48) CA1CA2CA12CA9POLB
SCHEMBL25074671 0.77 ABL1 (0.37) CA1CA2CA12CA9POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114901646-B Benzotriazine bisoxides and pharmaceutical compositions thereof 浙江瑞臻医药有限公司 2024-06-04 CN disclosed
WO-2023019912-A9 BENZOTRIAZINE DIOXIDE AND PHARMACEUTICAL COMPOSITION THEREOF 杭州瑞臻医药有限公司 2023-06-01 WO disclosed
WO-2023019912-A1 BENZOTRIAZINE DIOXIDE AND PHARMACEUTICAL COMPOSITION THEREOF 杭州瑞臻医药有限公司 2023-02-23 WO disclosed
CN-114901646-A Benzotriazine double oxide and pharmaceutical composition thereof 杭州瑞臻医药有限公司 2022-08-12 CN disclosed