Nimucitinib

Nimucitinib

SCHEMBL25254372

NC(=O)c1cnc(Nc2cccc(NC(=O)C3CCCNC3)c2)cc1NCc1cc(F)cc(F)c1

nearest known ligand 0.54

Full drug profile on Sugi Atlas →

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
AURKA O14965 2/20 0.54
AURKB Q96GD4 2/20 0.54
JAK3 P52333 7/20 0.49
IRAK4 Q9NWZ3 4/20 0.49
JAK2 O60674 2/20 0.49
JAK1 P23458 2/20 0.49
TYK2 P29597 2/20 0.49
RPS6KB1 P23443 1/20 0.48
CSF1R P07333 1/20 0.47
BTK Q06187 1/20 0.47
NTRK1 P04629 1/20 0.44
CDK9 P50750 9/20 0.44
F10 P00742 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Nimucitinib SCHEMBL25217505 1.00 AURKA (0.54) AURKAAURKBJAK3IRAK4JAK2
Nimucitinib SCHEMBL30431368 1.00 AURKA (0.54) AURKAAURKBJAK3IRAK4JAK2
Nimucitinib SCHEMBL25269469 1.00 AURKA (0.54) AURKAAURKBJAK3IRAK4JAK2
Nimucitinib SCHEMBL30431422 1.00 AURKA (0.54) AURKAAURKBJAK3IRAK4JAK2
SCHEMBL26173194 0.85 JAK3 (0.48) AURKAAURKBJAK3IRAK4JAK2
SCHEMBL12206906 0.85 JAK3 (0.63) AURKAAURKBJAK3IRAK4JAK2
SCHEMBL25260540 0.84 AURKA (0.43) AURKAAURKBNTRK1CDK9F10
Hydrochloric Acid SCHEMBL2484232 0.84 JAK3 (0.62) AURKAAURKBJAK3IRAK4JAK2
SCHEMBL2485627 0.83 JAK3 (0.53) AURKAJAK3IRAK4JAK2JAK1
Hydrochloric Acid SCHEMBL2484490 0.83 JAK3 (0.52) AURKAJAK3IRAK4JAK2JAK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023100918-A1 NOVEL NICOTINAMIDE COMPOUND AND USE THEREFOR 興和株式会社 2023-06-08 WO claimed
WO-2023100918-A1 NOVEL NICOTINAMIDE COMPOUND AND USE THEREFOR 興和株式会社 2023-06-08 WO disclosed
WO-2023100918-A1 NOVEL NICOTINAMIDE COMPOUND AND USE THEREFOR 興和株式会社 2023-06-08 WO disclosed