SCHEMBL25267697

SCHEMBL25267697

C[C@H]1NCCn2c(-c3ccc(F)c(F)c3)nnc21

nearest known ligand 0.51

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TACR3 P29371 8/20 0.51
TACR2 P21452 4/20 0.38
KCNH2 Q12809 4/20 0.37
TACR1 P25103 3/20 0.35
P2RX7 Q99572 1/20 0.35
GAA P10253 1/20 0.35
TSHR P16473 1/20 0.35
STAT3 P40763 1/20 0.34
DRD3 P35462 2/20 0.33
TP53 P04637 1/20 0.33
CREBBP Q92793 1/20 0.32
NOTUM Q6P988 1/20 0.32
PSEN1 P49768 1/20 0.32
PSEN2 P49810 1/20 0.32
APH1B Q8WW43 1/20 0.32
NCSTN Q92542 1/20 0.32
APH1A Q96BI3 1/20 0.32
PSENEN Q9NZ42 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL928992 0.80 TACR3 (0.50) TACR3GAATSHR
SCHEMBL25280034 0.80 TP53 (0.54) TACR3TACR2KCNH2TP53
SCHEMBL31055679 0.80 TP53 (0.54) TACR3TACR2KCNH2TP53
SCHEMBL25225767 0.80 TP53 (0.54) TACR3TACR2KCNH2TP53
SCHEMBL928185 0.79 TACR3 (0.57) TACR3P2RX7GAATSHR
SCHEMBL18417159 0.75 TACR3 (0.48) TACR3TSHRCREBBPNOTUM
SCHEMBL18417158 0.75 TACR3 (0.48) TACR3TSHRCREBBPNOTUM
SCHEMBL25219961 0.74 TACR3 (0.47) TACR3TACR2KCNH2TACR1
SCHEMBL25270063 0.74 TACR3 (0.47) TACR3TACR2KCNH2TACR1
SCHEMBL18916724 0.74 TACR3 (0.56) TACR3KCNH2GAATSHRTP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4190784-A1 NITROGEN-CONTAINING FUSED RING DERIVATIVE INHIBITOR, PREPARATION METHOD THEREFOR AND USE THEREOF Shanghai Hansoh Biomedical Co., Ltd. (CN) 2023-06-07 EP disclosed