SCHEMBL2529079

SCHEMBL2529079

CC(=O)COc1cc2cc(c1)C(=O)N[C@H]([C@H](O)CNC1(c3cc(C(C)(C)C)ccn3)CC1)Cc1cccc(c1)OCCCCO2

nearest known ligand 0.55

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 20/20 0.55
CTSD P07339 9/20 0.52
CTSE P14091 4/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2530320 0.96 BACE1 (0.51) BACE1CTSDCTSE
SCHEMBL2531242 0.86 BACE1 (0.67) BACE1CTSDCTSE
SCHEMBL2532272 0.85 BACE1 (0.71) BACE1CTSDCTSE
SCHEMBL2529797 0.85 BACE1 (0.64) BACE1CTSDCTSE
SCHEMBL2533578 0.84 BACE1 (0.71) BACE1CTSDCTSE
SCHEMBL2531265 0.83 BACE1 (0.63) BACE1CTSDCTSE
SCHEMBL2525909 0.83 BACE1 (0.80) BACE1CTSDCTSE
SCHEMBL4872628 0.82 BACE1 (0.47) BACE1CTSDCTSE
SCHEMBL2534353 0.82 BACE1 (0.63) BACE1CTSDCTSE
SCHEMBL2526933 0.80 BACE1 (0.66) BACE1CTSDCTSE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8039455-B2 Macrocyclic compounds useful as BACE inhibitors NOVARTIS AG (CH) 2011-10-18 US claimed