SCHEMBL25293100

SCHEMBL25293100

CN1CC=C(c2c[nH]c3c(Cl)cccc23)C1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 2/20 0.49
SLC6A4 P31645 3/20 0.46
KDM4E B2RXH2 1/20 0.46
LMNA P02545 1/20 0.46
POLB P06746 1/20 0.46
HTR1A P08908 1/20 0.46
ALOX15 P16050 1/20 0.46
HTR6 P50406 1/20 0.46
HSD17B10 Q99714 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
AR P10275 2/20 0.43
DYRK1A Q13627 3/20 0.41
PRKCB P05771 1/20 0.41
PRKCA P17252 1/20 0.41
PRKCH P24723 1/20 0.41
PRKCE Q02156 1/20 0.41
PRKCQ Q04759 1/20 0.41
PRKCD Q05655 1/20 0.41
NR4A2 P43354 1/20 0.39
RIPK1 Q13546 3/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30548044 1.00 HTR2A (0.49) HTR2ASLC6A4KDM4ELMNAPOLB
SCHEMBL7866280 0.86 SLC6A4 (0.64) SLC6A4KDM4ELMNAPOLBHTR1A
SCHEMBL30548025 0.86 HTR2A (0.66) HTR2AARPRKCBPRKCAPRKCH
SCHEMBL25288178 0.86 HTR2A (0.66) HTR2AARPRKCBPRKCAPRKCH
SCHEMBL25286351 0.76 HTR2A (0.48) HTR2A
SCHEMBL25290977 0.76 KDM4E (0.54) HTR2ASLC6A4KDM4ELMNAPOLB
SCHEMBL25248306 0.76 HTR2A (0.47) HTR2AKDM4ELMNAALOX15AR
SCHEMBL25293430 0.74 CHEK1 (0.45) HTR2ASLC6A4KDM4ELMNAPOLB
SCHEMBL16801563 0.74 MAPT (0.50) SLC6A4KDM4ELMNAPOLBHTR1A
SCHEMBL25290621 0.72 AR (0.46) HTR2ASLC6A4KDM4EALOX15HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023114472-A1 HETEROCYCLIC COMPOUNDS AS 5HT2A BIASED AGONISTS ICAHN SCHOOL OF MEDICINE AT MOUNT SINAI (US) 2023-06-22 WO disclosed
WO-2023114472-A1 HETEROCYCLIC COMPOUNDS AS 5HT2A BIASED AGONISTS ICAHN SCHOOL OF MEDICINE AT MOUNT SINAI (US) 2023-06-22 WO disclosed