SCHEMBL2529792

SCHEMBL2529792

CC(C)(C)C1CCC(Oc2ccc3cc([C@@](C)(N)CO)ccc3c2)CC1.[Fe]

nearest known ligand 0.42

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 5/20 0.42
ENPP2 Q13822 3/20 0.36
TRPV1 Q8NER1 1/20 0.35
SRC P12931 1/20 0.35
S1PR5 Q9H228 3/20 0.34
CYP19A1 P11511 1/20 0.34
ABL1 P00519 1/20 0.34
HRH3 Q9Y5N1 1/20 0.34
MAPT P10636 1/20 0.33
NPC1L1 Q9UHC9 1/20 0.33
MAOA P21397 1/20 0.33
MAOB P27338 1/20 0.33
SCN10A Q9Y5Y9 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2775755 0.99 KCNH2 (0.43) KCNH2ENPP2TRPV1SRCS1PR5
SCHEMBL2775752 0.99 KCNH2 (0.43) KCNH2ENPP2TRPV1SRCS1PR5
SCHEMBL2777056 0.99 KCNH2 (0.43) KCNH2ENPP2TRPV1SRCS1PR5
SCHEMBL2452603 0.99 KCNH2 (0.43) KCNH2ENPP2TRPV1SRCS1PR5
SCHEMBL2777408 0.91 KCNH2 (0.41) KCNH2ENPP2TRPV1SRCS1PR5
SCHEMBL2777405 0.91 KCNH2 (0.41) KCNH2ENPP2TRPV1SRCS1PR5
SCHEMBL2451591 0.89 KCNH2 (0.41) KCNH2TRPV1SRCABL1HRH3
SCHEMBL2452030 0.89 KCNH2 (0.41) KCNH2ENPP2SRCABL1HRH3
SCHEMBL2452283 0.89 KCNH2 (0.41) KCNH2ENPP2SRCABL1HRH3
SCHEMBL2451587 0.89 KCNH2 (0.41) KCNH2TRPV1SRCABL1HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2364088-A1 BICYCLIC ARYL SPHINGOSINE 1-PHOSPHATE ANALOGS Biogen Idec MA Inc. (US) 2011-09-14 EP disclosed
WO-2010051030-A1 BICYCLIC ARYL SPHINGOSINE 1-PHOSPHATE ANALOGS BIOGEN IDEC MA INC. (US) 2010-05-06 WO disclosed