SCHEMBL25305296

SCHEMBL25305296

O=C(N1CCOCC1)N1CCc2cc(Cl)cc(C3COCCN3)c2C1

nearest known ligand 0.36

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 9/20 0.36
L3MBTL1 Q9Y468 1/20 0.33
KCNK3 O14649 1/20 0.33
KIF11 P52732 1/20 0.32
DRD2 P14416 1/20 0.32
DRD3 P35462 1/20 0.32
HRH3 Q9Y5N1 1/20 0.32
OPRM1 P35372 1/20 0.31
KDM4E B2RXH2 1/20 0.31
MEN1 O00255 1/20 0.31
GAA P10253 1/20 0.31
TSHR P16473 1/20 0.31
KMT2A Q03164 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25305291 1.00 AKR1C3 (0.36) AKR1C3L3MBTL1KCNK3KIF11DRD2
SCHEMBL30491431 0.92 AKR1C3 (0.33) AKR1C3HRH3TSHR
SCHEMBL30491427 0.88 PRMT5 (0.33) DRD2DRD3
SCHEMBL30491502 0.88 GLRA1 (0.33) DRD2DRD3
SCHEMBL30068848 0.88 AKR1C3 (0.36) AKR1C3L3MBTL1KIF11DRD2DRD3
SCHEMBL30491452 0.88 BAZ2B (0.39) KCNK3
SCHEMBL30491388 0.88 GRM5 (0.34) DRD2DRD3MEN1TSHRKMT2A
SCHEMBL25306100 0.87
SCHEMBL25306095 0.87
SCHEMBL25253225 0.87 GRM5 (0.30)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023131122-A1 FUSED RING-SUBSTITUTED SIX-MEMBERED HETEROCYCLIC COMPOUND, AND PREPARATION METHOD THEREFOR AND USE THEREOF 劲方医药科技(上海)有限公司 2023-07-13 WO disclosed