SCHEMBL2531645

SCHEMBL2531645

COCc1cc2cc(c1)C(=O)N[C@H]([C@H](O)CNC1(c3cc(C(C)C)ccn3)CC1)Cc1cccc(c1)CCCCN2

nearest known ligand 0.68

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 20/20 0.68
CTSD P07339 6/20 0.68
CTSE P14091 4/20 0.68

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2532830 0.91 BACE1 (0.66) BACE1CTSDCTSE
SCHEMBL2531362 0.91 BACE1 (0.83) BACE1CTSDCTSE
SCHEMBL2533816 0.90 BACE1 (0.82) BACE1CTSDCTSE
SCHEMBL2528412 0.88 BACE1 (0.57) BACE1CTSDCTSE
SCHEMBL2528417 0.87 BACE1 (0.56) BACE1CTSDCTSE
SCHEMBL4880824 0.86 BACE1 (0.68) BACE1CTSDCTSE
SCHEMBL2525932 0.84 BACE1 (0.49) BACE1CTSDCTSE
SCHEMBL4878120 0.83 BACE1 (0.81) BACE1CTSDCTSE
SCHEMBL2525909 0.82 BACE1 (0.80) BACE1CTSDCTSE
SCHEMBL2529506 0.81 BACE1 (1.00) BACE1CTSDCTSE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8039455-B2 Macrocyclic compounds useful as BACE inhibitors NOVARTIS AG (CH) 2011-10-18 US claimed
US-8039455-B2 Macrocyclic compounds useful as BACE inhibitors NOVARTIS AG (CH) 2011-10-18 US disclosed