SCHEMBL25326552

SCHEMBL25326552

CCOC(=O)c1cc(-c2ccnc(Nc3cc(OC)c(OC)c(OC)c3)n2)nn1C

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SYK P43405 16/20 0.63
FLT3 P36888 12/20 0.53
JAK2 O60674 10/20 0.53
CDK2 P24941 3/20 0.52
AURKA O14965 2/20 0.52
CDK1 P06493 2/20 0.52
CDK7 P50613 2/20 0.52
CDK9 P50750 2/20 0.52
AURKB Q96GD4 2/20 0.52
CDK4 P11802 1/20 0.52
LYN P07948 1/20 0.52
PRKCB P05771 2/20 0.52
ZAP70 P43403 2/20 0.52
PRKD3 O94806 1/20 0.52
PRKCG P05129 1/20 0.52
LCK P06239 1/20 0.52
PRKCA P17252 1/20 0.52
PRKCH P24723 1/20 0.52
PRKCI P41743 1/20 0.52
PRKCE Q02156 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25330513 0.91 SYK (0.63) SYKFLT3JAK2LYNPRKCB
SCHEMBL25326858 0.89 SYK (0.62) SYKFLT3JAK2LYNPRKCB
SCHEMBL25327751 0.87 SYK (0.66) SYKFLT3JAK2CDK2AURKA
SCHEMBL29492416 0.87 SYK (0.69) SYKFLT3JAK2LYN
SCHEMBL25329262 0.87 SYK (0.69) SYKFLT3JAK2LYN
SCHEMBL25328787 0.85 SYK (0.60) SYKFLT3JAK2LYN
SCHEMBL25329120 0.85 SYK (0.60) SYKFLT3JAK2LYN
SCHEMBL25328122 0.84 SYK (0.56) SYKFLT3JAK2LYNPRKCB
SCHEMBL25328086 0.84 SYK (0.64) SYKFLT3JAK2CDK2AURKA
SCHEMBL25327260 0.83 SYK (0.53) SYKFLT3JAK2LYNPRKCB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240285621-A1 PYRAZOLYL-PYRIMIDINE DERIVATIVES AS KINASE INHIBITORS NERVIANO MEDICAL SCIENCES S.R.L. (IT) 2024-08-29 US disclosed
EP-4217354-A1 PYRAZOLYL-PYRIMIDINE DERIVATIVES AS KINASE INHIBITORS Nerviano Medical Sciences S.r.l. (IT) 2023-08-02 EP disclosed
CN-116323595-A Pyrazolyl-pyrimidine derivatives as kinase inhibitors 内尔维亚诺医疗科学公司 2023-06-23 CN disclosed
WO-2022063646-A1 PYRAZOLYL-PYRIMIDINE DERIVATIVES AS KINASE INHIBITORS NERVIANO MEDICAL SCIENCES S.R.L. (IT) 2022-03-31 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240285621-A1 PYRAZOLYL-PYRIMIDINE DERIVATIVES AS KINASE INHIBITORS SYK, LCK, BTK SYK 1/4885FLT3 28/4885JAK2 12/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.