SCHEMBL2533071

SCHEMBL2533071

O=C(c1ccc(B(O)O)cc1)N1CCOCC1.OBO

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PHGDH O43175 1/20 0.59
HPGD P15428 6/20 0.56
AKR1C3 P42330 1/20 0.54
TSHR P16473 1/20 0.53
L3MBTL1 Q9Y468 3/20 0.52
ALDH1A1 P00352 3/20 0.52
SMN1; SMN2 Q16637 2/20 0.52
MAPK1 P28482 1/20 0.52
KDM4E B2RXH2 1/20 0.52
MAPT P10636 1/20 0.52
HTT P42858 1/20 0.52
POLB P06746 1/20 0.51
DNMT1 P26358 1/20 0.51
PTPN7 P35236 1/20 0.51
KMT2A Q03164 1/20 0.51
TDP1 Q9NUW8 1/20 0.51
PKM P14618 1/20 0.51
MLYCD O95822 1/20 0.51
EPHX2 P34913 1/20 0.49
L3MBTL3 Q96JM7 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL109091 0.95 PHGDH (0.65) PHGDHHPGDAKR1C3TSHRL3MBTL1
SCHEMBL2040124 0.87 PHGDH (0.55) PHGDHHPGDAKR1C3TSHRL3MBTL1
SCHEMBL29950978 0.83 HPGD (0.57) HPGDALDH1A1SMN1; SMN2MAPK1HTT
SCHEMBL10720943 0.83 PHGDH (0.81) PHGDHHPGDAKR1C3TSHRL3MBTL1
SCHEMBL950365 0.80 HPGD (0.64) HPGDTSHRALDH1A1SMN1; SMN2MAPK1
SCHEMBL204078 0.80 HPGD (0.70) HPGDTSHRL3MBTL1ALDH1A1MAPK1
SCHEMBL12960648 0.79 PHGDH (0.65) PHGDHHPGDAKR1C3TSHRL3MBTL1
SCHEMBL258027 0.78 HPGD (0.74) HPGDTSHRL3MBTL1ALDH1A1MAPK1
SCHEMBL28296651 0.78 HPGD (0.86) PHGDHHPGDAKR1C3TSHRL3MBTL1
SCHEMBL8123 0.77 TSHR (0.60) HPGDTSHRL3MBTL1ALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8034940-B2 Modulators of glucocorticoid receptor, AP-1, and/or NF-κB activity and use thereof BRISTOL-MYERS SQUIBB COMPANY (US) 2011-10-11 US disclosed