SCHEMBL2533386

SCHEMBL2533386

CN1Cc2cc(Cl)ccc2-n2c(nnc2C2CCC(Oc3ccc(F)cn3)CC2)C1.Fc1ccc(OC2CCC(c3nnc4n3-c3ccc(Cl)cc3CNC4)CC2)nc1

nearest known ligand 0.68

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
AVPR1A P37288 20/20 0.68
KCNH2 Q12809 9/20 0.68
AVPR2 P30518 6/20 0.68

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3331544 0.94 AVPR1A (0.76) AVPR1AKCNH2AVPR2
SCHEMBL3331550 0.94 AVPR1A (0.76) AVPR1AKCNH2AVPR2
SCHEMBL3330990 0.93 AVPR1A (0.62) AVPR1AKCNH2AVPR2
SCHEMBL2469534 0.93 AVPR1A (0.62) AVPR1AKCNH2AVPR2
SCHEMBL3329662 0.88 AVPR1A (0.80) AVPR1AKCNH2AVPR2
SCHEMBL2475500 0.88 AVPR1A (0.80) AVPR1AKCNH2AVPR2
SCHEMBL15234269 0.87 AVPR1A (0.61) AVPR1AKCNH2AVPR2
SCHEMBL11934674 0.87 AVPR1A (0.61) AVPR1AKCNH2AVPR2
Hydrochloric Acid SCHEMBL3330082 0.86 AVPR1A (0.60) AVPR1AKCNH2AVPR2
Hydrochloric Acid SCHEMBL2475011 0.86 AVPR1A (0.60) AVPR1AKCNH2AVPR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2370441-A1 ARYLCYCLOHEXYLETHERS OF DIHYDROTETRAAZABENZOAZULENES FOR USE AS VASOPRESSIN VIA RECEPTOR ANTAGONISTS F. Hoffmann-La Roche AG (CH) 2011-10-05 EP claimed