SCHEMBL2541013

SCHEMBL2541013

CC(Oc1cc(-c2cnc3ccc(CN(C)C)nn23)sc1C(N)=O)c1ccccc1Cl

nearest known ligand 0.68

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
PLK1 P53350 20/20 0.68
PLK3 Q9H4B4 1/20 0.51
CYP3A4 P08684 1/20 0.51
CYP2C9 P11712 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2541011 1.00 PLK1 (0.68) PLK1PLK3CYP3A4CYP2C9
SCHEMBL2517944 0.92 PLK1 (0.74) PLK1
SCHEMBL2517941 0.92 PLK1 (0.74) PLK1
SCHEMBL2521625 0.89 PLK1 (0.72) PLK1
SCHEMBL2521623 0.89 PLK1 (0.72) PLK1
SCHEMBL2520767 0.87 PLK1 (0.84) PLK1
SCHEMBL2520809 0.86 PLK1 (0.69) PLK1
SCHEMBL1370934 0.83 PLK1 (0.75) PLK1
SCHEMBL2521641 0.83 PLK1 (0.80) PLK1
SCHEMBL2521637 0.83 PLK1 (0.80) PLK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8030327-B2 3-[1-(2-chlorophenyl)ethoxy]-5-imidazo[1,2-a]pyridin-3-ylthiophene-2-carboxyamide; polo like kinase inhibitor; antitumor and anticarcinogenic agent; mitotic phase (M phase) of the cell cycle MDS K.K. (JP) 2011-10-04 US disclosed
US-20080103136-A1 Novel Fused Imidazole Derivative MSD K.K. (JP) 2008-05-01 US disclosed
EP-1813613-A1 NOVEL FUSED IMIDAZOLE DERIVATIVE BANYU PHARMACEUTICAL CO., LTD. (JP) 2007-08-01 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080103136-A1 Novel Fused Imidazole Derivative HRH4, H1-4, H1-3 PLK1 4301/4885PLK3 3835/4885CYP3A4 26/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.