SCHEMBL2541609

SCHEMBL2541609

CCc1cc(Nc2nccc3[nH]nc(OCCOS(C)(=O)=O)c23)ccc1OCc1ccccn1

nearest known ligand 0.51

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ERBB2 P04626 18/20 0.51
EGFR P00533 16/20 0.51
GRM4 Q14833 1/20 0.39
ERBB3 P21860 1/20 0.38
ERBB4 Q15303 1/20 0.38
KCNH2 Q12809 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2544438 0.91 ERBB2 (0.55) ERBB2EGFR
SCHEMBL1406489 0.89 ERBB2 (0.63) ERBB2EGFRERBB3ERBB4
SCHEMBL2515600 0.83 EGFR (0.68) ERBB2EGFRGRM4
SCHEMBL1406571 0.80 ERBB2 (0.67) ERBB2EGFR
SCHEMBL2515689 0.79 ERBB2 (0.55) ERBB2EGFRKCNH2
SCHEMBL2516578 0.78 EGFR (0.60) ERBB2EGFRGRM4ERBB3ERBB4
SCHEMBL2524606 0.78 ERBB2 (0.65) ERBB2EGFR
SCHEMBL2514377 0.78 ERBB2 (0.67) ERBB2EGFRGRM4ERBB3ERBB4
SCHEMBL2518693 0.78 ERBB2 (0.67) ERBB2EGFRGRM4ERBB3ERBB4
SCHEMBL2522405 0.78 EGFR (0.56) ERBB2EGFRERBB4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1838712-B8 PYRAZOLOPYRIMIDINE COMPOUNDS AS ANTITUMOR AGENTS ASTRAZENECA AB (SE) 2011-10-12 EP disclosed
EP-1838712-A1 PYRAZOLOPYRIMIDINE COMPOUNDS AS ANTITUMOR AGENTS AstraZeneca AB (SE) 2007-10-03 EP disclosed
WO-2006064196-A1 PYRAZOLOPYRIMIDINE COMPOUNDS AS ANTITUMOR AGENTS ASTRAZENECA AB (SE) 2006-06-22 WO disclosed