SCHEMBL25427809

SCHEMBL25427809

O=C1CCC(N2Cc3cc(Br)cc(OC(F)F)c3C2=O)C(=O)N1

nearest known ligand 0.48

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CRBN Q96SW2 16/20 0.48
IKZF2 Q9UKS7 3/20 0.41
CSNK1A1 P48729 2/20 0.41
ESR1 P03372 1/20 0.41
DDB1 Q16531 1/20 0.41
SALL4 Q9UJQ4 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24717680 0.86 CRBN (0.51) CRBNIKZF2CSNK1A1DDB1
SCHEMBL21477242 0.83 CRBN (0.65) CRBNDDB1
SCHEMBL20231758 0.82 ESR1 (0.48) CRBNESR1DDB1
SCHEMBL24717677 0.82 CRBN (0.54) CRBNIKZF2DDB1
SCHEMBL26184312 0.82 CRBN (0.56) CRBNIKZF2DDB1
SCHEMBL30270743 0.82 CRBN (0.56) CRBNIKZF2CSNK1A1DDB1
SCHEMBL25012254 0.82 CRBN (0.56) CRBNIKZF2CSNK1A1DDB1
SCHEMBL25010116 0.80 CRBN (0.54) CRBNIKZF2DDB1
SCHEMBL25010168 0.80 CRBN (0.54) CRBNIKZF2DDB1
SCHEMBL25010291 0.79 CRBN (0.51) CRBNIKZF2DDB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4466260-A1 COMPOUNDS AND THEIR USE IN TREATING CANCER Astrazeneca AB (SE) 2024-11-27 EP disclosed
CN-118574821-A Compounds and their use in the treatment of cancer 阿斯利康(瑞典)有限公司 2024-08-30 CN disclosed
WO-2023139199-A1 COMPOUNDS AND THEIR USE IN TREATING CANCER ASTRAZENECA AB (SE) 2023-07-27 WO disclosed
WO-2023139199-A1 COMPOUNDS AND THEIR USE IN TREATING CANCER ASTRAZENECA AB (SE) 2023-07-27 WO disclosed