SCHEMBL25435280

SCHEMBL25435280

COCOc1cc(-c2ncc3c(N4CCC(N5CCCC5)CC4)nc(OC[C@@]45CCCN4C[C@H](F)C5)nc3c2F)c2c(C#C[Si](C(C)C)(C(C)C)C(C)C)c(F)ccc2c1

nearest known ligand 0.57

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
KRAS P01116 20/20 0.57
MAPK3 P27361 1/20 0.57
MAPK1 P28482 1/20 0.57
RAF1 P04049 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25404453 0.95 KRAS (0.58) KRASMAPK3MAPK1RAF1
SCHEMBL29341154 0.93 KRAS (0.57) KRASMAPK3MAPK1RAF1
SCHEMBL25401862 0.92 KRAS (0.58) KRASMAPK3MAPK1RAF1
SCHEMBL25402031 0.92 KRAS (0.57) KRASMAPK3MAPK1RAF1
SCHEMBL31170188 0.92 KRAS (0.58) KRASMAPK3MAPK1RAF1
SCHEMBL25437473 0.91 KRAS (0.68) KRASMAPK3MAPK1RAF1
SCHEMBL29679922 0.91 KRAS (0.59) KRASMAPK3MAPK1RAF1
SCHEMBL29680017 0.91 KRAS (0.59) KRASMAPK3MAPK1RAF1
SCHEMBL29049543 0.91 KRAS (0.56) KRASMAPK3MAPK1RAF1
SCHEMBL27117552 0.91 KRAS (0.55) KRASMAPK3MAPK1RAF1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023138583-A1 HETEROCYCLIC COMPOUND, PHARMACEUTICAL COMPOSITION AND USE THEREOF 上海湃隆生物科技有限公司 2023-07-27 WO disclosed