SCHEMBL25437151

SCHEMBL25437151

CNC(=O)c1cc(CN(CCC2CC3CN(c4ccc(Br)cn4)CC3C2)C(=O)O)on1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM4 P08173 1/20 0.34
ACACB O00763 1/20 0.33
NPC1 O15118 2/20 0.32
RAB9A P51151 2/20 0.32
AKR1C3 P42330 1/20 0.31
PDE10A Q9Y233 1/20 0.31
LMNA P02545 2/20 0.31
HPGD P15428 2/20 0.31
SMN1; SMN2 Q16637 2/20 0.31
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
HDAC3 O15379 1/20 0.31
HDAC4 P56524 1/20 0.31
HDAC1 Q13547 1/20 0.31
HDAC7 Q8WUI4 1/20 0.31
HDAC2 Q92769 1/20 0.31
HDAC10 Q969S8 1/20 0.31
HDAC11 Q96DB2 1/20 0.31
HDAC8 Q9BY41 1/20 0.31
HDAC6 Q9UBN7 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8513298 1.00 CHRM4 (0.34) CHRM4ACACBNPC1RAB9AAKR1C3
SCHEMBL8513303 1.00 CHRM4 (0.34) CHRM4ACACBNPC1RAB9AAKR1C3
SCHEMBL8512856 0.89 AKR1C3 (0.32) CHRM4ACACBAKR1C3PDE10A
SCHEMBL25435089 0.89 AKR1C3 (0.32) CHRM4ACACBAKR1C3PDE10A
SCHEMBL8512859 0.89 AKR1C3 (0.32) CHRM4ACACBAKR1C3PDE10A
SCHEMBL25437153 0.82 ACACB (0.35) CHRM4ACACBAKR1C3PDE10AHDAC3
SCHEMBL8510068 0.74 PDE10A (0.42) RAB9APDE10AHDAC3HDAC4HDAC1
SCHEMBL8510075 0.74 PDE10A (0.42) RAB9APDE10AHDAC3HDAC4HDAC1
SCHEMBL9994507 0.73 CHRM4 (0.33) CHRM4NPC1RAB9AAKR1C3LMNA
SCHEMBL25435091 0.72 ACACB (0.34) CHRM4ACACBNPC1RAB9AAKR1C3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3856735-B1 FUSED BICYCLIC HETEROCYCLES AS THERAPEUTIC AGENTS UNIV NEW YORK (US) 2023-09-06 EP claimed