SCHEMBL2545372

SCHEMBL2545372

CC(=O)c1cccc(-c2ccc(C3=N[C@@H](C(C)C(=O)O)c4nnc(CO)n4-c4sc(C)c(C)c43)cc2)c1

nearest known ligand 0.44

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 20/20 0.44
DNER Q8NFT8 1/20 0.40
BRDT Q58F21 4/20 0.39
BRD2 P25440 3/20 0.39
ADORA3 P0DMS8 1/20 0.39
TSPO P30536 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2534315 0.90 BRD4 (0.52) BRD4DNERBRDTBRD2ADORA3
SCHEMBL2543043 0.88 BRD4 (0.58) BRD4DNERBRDT
SCHEMBL2543487 0.86 BRD4 (0.51) BRD4DNERBRDT
SCHEMBL3211715 0.86 BRD4 (0.59) BRD4DNERBRDTBRD2ADORA3
SCHEMBL2545756 0.85 BRD4 (0.50) BRD4DNERBRDTBRD2ADORA3
SCHEMBL2537131 0.83 BRD4 (0.52) BRD4DNERBRDTBRD2ADORA3
SCHEMBL2542552 0.83 BRD4 (0.53) BRD4DNERBRDTBRD2ADORA3
SCHEMBL2541446 0.83 BRD4 (0.52) BRD4DNERBRDTBRD2ADORA3
SCHEMBL2541274 0.81 BRD4 (0.51) BRD4DNERBRDT
SCHEMBL2540559 0.81 BRD4 (0.46) BRD4BRDTADORA3TSPO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8044042-B2 Thienotriazolodiazepine compound and medicinal use thereof MITSUBISHI TANABE PHARMA CORPORATION (JP) 2011-10-25 US disclosed