SCHEMBL2550839

SCHEMBL2550839

COc1ccc2[nH]c(=O)c3scc(C4=CCCCC4)c3c2c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.43
HTT P42858 3/20 0.43
NPSR1 Q6W5P4 2/20 0.43
CYP1A2 P05177 2/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
PPARG P37231 1/20 0.43
NCOA2 Q15596 1/20 0.43
NCOA1 Q15788 1/20 0.43
RXFP1 Q9HBX9 1/20 0.43
NCOA3 Q9Y6Q9 1/20 0.43
PDGFRB P09619 1/20 0.40
DYRK1A Q13627 2/20 0.39
KDR P35968 1/20 0.39
MAOA P21397 1/20 0.39
ACHE P22303 1/20 0.39
MAOB P27338 1/20 0.39
BACE1 P56817 1/20 0.39
ALDH1A1 P00352 6/20 0.38
KDM4E B2RXH2 5/20 0.38
MEN1 O00255 4/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2546499 0.84 PARP1 (0.40) PARP1DYRK1AMEN1KMT2ACSF1R
SCHEMBL2545355 0.68 NEK1 (0.60)
SCHEMBL2549121 0.67 KDM4E (0.57) PARP1HTTNPSR1CYP1A2SMN1; SMN2
SCHEMBL2553660 0.65 PARP1 (0.69) PARP1CYP1A2KDRALDH1A1KDM4E
SCHEMBL3148434 0.65 NPC1 (0.52) HTTNPSR1SMN1; SMN2ACHEALDH1A1
SCHEMBL1516053 0.64 NPC1 (0.51) CYP1A2ACHEALDH1A1KMT2ATSHR
SCHEMBL2547281 0.63 HTT (0.57) PARP1HTTNPSR1CYP1A2SMN1; SMN2
Hydrochloric Acid SCHEMBL2367094 0.62 PARP1 (0.97) PARP1KDR
SCHEMBL3148438 0.62 NPC1 (0.49) HTTALDH1A1KDM4EMEN1KMT2A
SCHEMBL2550137 0.62 CSNK2A1 (0.51) PARP1HTTNPSR1CYP1A2SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2552206-A1 TRYCYCLIC COMPOUNDS AND PBK INHIBITORS CONTAINING THE SAME OncoTherapy Science, Inc. (JP) 2013-02-06 EP disclosed
WO-2011123419-A1 TRYCYCLIC COMPOUNDS AND PBK INHIBITORS CONTAINING THE SAME ONCOTHERAPY SCIENCE, INC. (JP) 2011-10-06 WO disclosed